EP 1851542 B1 20100414 - USE OF THIOPEPTOLIDES FOR DETERMINING THE ACTIVITY OF ADAMTS PROTEASES
Title (en)
USE OF THIOPEPTOLIDES FOR DETERMINING THE ACTIVITY OF ADAMTS PROTEASES
Title (de)
VERWENDUNG VON THIOPEPTOLIDEN ZUR AKTIVITÄTSBESTIMMUNG VON ADAM-TS PROTEASEN
Title (fr)
UTILISATION DE THIOPEPTOLIDES POUR DETECTER L'ACTIVITE DE PROTEASES ADAM-TS
Publication
Application
Priority
- EP 2006001184 W 20060210
- DE 102005005972 A 20050209
Abstract (en)
[origin: US2009149332A1] The invention concerns the use of thiopeptolides of formula R-(Xaa)n-Pro-X-Gly-S-Y-Z-Gly-(Xaa)m-R1 (I) as substrate for determining the activity of ADAMTS proteases, and a method for finding an ADAMTS protease modulator, more particularly an inhibitor.
IPC 8 full level
G01N 33/50 (2006.01)
CPC (source: EP KR US)
A61P 7/02 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07K 1/06 (2013.01 - KR); C12Q 1/37 (2013.01 - EP US); G01N 2500/00 (2013.01 - EP US); G01N 2800/102 (2013.01 - EP US); G01N 2800/105 (2013.01 - EP US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
US 2009149332 A1 20090611; AT E464563 T1 20100415; AU 2006220096 A1 20060908; BR PI0607059 A2 20090804; CA 2597862 A1 20060908; CN 101115993 A 20080130; DE 102005005972 A1 20060817; DE 502006006695 D1 20100527; EP 1851542 A1 20071107; EP 1851542 B1 20100414; IL 184769 A0 20071203; JP 2008543273 A 20081204; KR 20070120091 A 20071221; MX 2007009380 A 20070816; WO 2006092203 A1 20060908
DOCDB simple family (application)
US 81493606 A 20060210; AT 06706814 T 20060210; AU 2006220096 A 20060210; BR PI0607059 A 20060210; CA 2597862 A 20060210; CN 200680004289 A 20060210; DE 102005005972 A 20050209; DE 502006006695 T 20060210; EP 06706814 A 20060210; EP 2006001184 W 20060210; IL 18476907 A 20070722; JP 2007554503 A 20060210; KR 20077017908 A 20070802; MX 2007009380 A 20060210