EP 1857114 A1 20071121 - PARTICLE AND PREPARATION CONTAINING THE PARTICLE
Title (en)
PARTICLE AND PREPARATION CONTAINING THE PARTICLE
Title (de)
TEILCHEN UND DIESES TEILCHEN ENTHALTENDE ZUBEREITUNG
Title (fr)
PARTICULE ET PREPARATION LA CONTENANT
Publication
Application
Priority
- JP 2006304506 W 20060308
- JP 2005066158 A 20050309
Abstract (en)
The present invention relates to a particle having a mean particle size of 0.01 to 20 µm, containing tert-butyl (4R)-4-{[((1R)-2-[(1-benzylpiperidin-4-yl)amino]-1-{[(cyclohexylmethyl)thio]methyl}-2-oxoethyl)amino]carbonyl}-1,3-thiazolidine-3-carboxylate. A preparation containing the particle is excellent in pulmonary delivery through inhalation and is easy to handle because of excellent dispersibility of the particle, and thus the present compound can be used as a pulmonary preparation.
IPC 8 full level
A61K 38/00 (2006.01); A61K 9/72 (2006.01); A61K 47/24 (2006.01); A61K 47/26 (2006.01); A61K 47/38 (2006.01); A61P 29/00 (2006.01)
CPC (source: EP KR US)
A61K 9/00 (2013.01 - KR); A61K 9/0075 (2013.01 - EP US); A61K 38/00 (2013.01 - KR); A61P 25/04 (2017.12 - EP); A61P 29/00 (2017.12 - EP); C07D 417/12 (2013.01 - KR); A61K 9/1623 (2013.01 - EP US); A61K 9/1652 (2013.01 - EP US); Y10T 428/13 (2015.01 - EP US); Y10T 428/2982 (2015.01 - EP US)
Citation (search report)
See references of WO 2006095788A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
EP 1857114 A1 20071121; AU 2006221364 A1 20060914; BR PI0608844 A2 20100202; CA 2602007 A1 20060914; CN 101171023 A 20080430; IL 185590 A0 20080106; JP WO2006095788 A1 20080814; KR 20070110418 A 20071116; NO 20074505 L 20071210; RU 2007137121 A 20090420; US 2009022915 A1 20090122; WO 2006095788 A1 20060914; ZA 200707436 B 20090826
DOCDB simple family (application)
EP 06728775 A 20060308; AU 2006221364 A 20060308; BR PI0608844 A 20060308; CA 2602007 A 20060308; CN 200680016009 A 20060308; IL 18559007 A 20070829; JP 2006304506 W 20060308; JP 2007507162 A 20060308; KR 20077022785 A 20071005; NO 20074505 A 20070905; RU 2007137121 A 20060308; US 90809106 A 20060308; ZA 200707436 A 20070830