EP 1858850 B1 20150121 - PROCESS FOR THE PREPARATION OF OPIOID MODULATORS
Title (en)
PROCESS FOR THE PREPARATION OF OPIOID MODULATORS
Title (de)
HERSTELLUNGSVERFAHREN FÜR OPIOIDMODULATOREN
Title (fr)
PROCEDE POUR PREPARER DES MODULATEURS OPIOIDES
Publication
Application
Priority
- US 2006008450 W 20060306
- US 66178405 P 20050314
Abstract (en)
[origin: US2006211861A1] The present invention is directed to novel processes for the preparation of opioid modulators (agonists and antagonists) and intermediates in their synthesis. The opioid modulators are useful for the treatment and prevention of as pain and gastrointestinal disorders.
IPC 8 full level
C07D 233/61 (2006.01); C07D 233/64 (2006.01); C07D 401/04 (2006.01)
CPC (source: EP KR NO US)
A61P 1/00 (2017.12 - EP); A61P 1/04 (2017.12 - EP); A61P 1/10 (2017.12 - EP); A61P 1/12 (2017.12 - EP); A61P 25/04 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07C 233/11 (2013.01 - KR); C07C 237/14 (2013.01 - KR); C07D 211/60 (2013.01 - KR); C07D 217/26 (2013.01 - KR); C07D 233/61 (2013.01 - EP NO US); C07D 233/64 (2013.01 - EP NO US); C07D 401/04 (2013.01 - EP NO US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA HR MK YU
DOCDB simple family (publication)
US 2006211861 A1 20060921; AR 053170 A1 20070425; AR 054745 A1 20070711; AU 2006223394 A1 20060921; AU 2006223394 B2 20121018; AU 2006223482 A1 20060921; BR PI0607792 A2 20090613; BR PI0607793 A2 20090613; CA 2601481 A1 20060921; CA 2601481 C 20131112; CA 2601674 A1 20060921; CN 101175725 A 20080507; CN 101175725 B 20110202; CN 101175726 A 20080507; CR 9438 A 20080909; CY 1116104 T1 20170208; DK 1858850 T3 20150209; EA 014366 B1 20101029; EA 015512 B1 20110830; EA 200701978 A1 20080428; EA 200701979 A1 20080428; EP 1858850 A2 20071128; EP 1858850 B1 20150121; EP 1863764 A1 20071212; ES 2535048 T3 20150504; HR P20150417 T1 20150925; HU E024912 T2 20160229; IL 185972 A0 20080106; IL 185972 A 20130731; IL 185974 A0 20080106; IL 209402 A0 20110131; IL 209402 A 20150630; JP 2008533141 A 20080821; JP 2008533143 A 20080821; JP 2013234192 A 20131121; JP 5384933 B2 20140108; JP 5802242 B2 20151028; KR 101280929 B1 20130701; KR 20070112255 A 20071122; KR 20070116067 A 20071206; ME 02110 B 20151020; MX 2007011409 A 20080222; MX 2007011412 A 20080222; MY 145333 A 20120131; NI 200700237 A 20080625; NO 20075268 L 20071210; NO 20075269 L 20071210; NO 340604 B1 20170515; NZ 590570 A 20120629; PL 1858850 T3 20150630; PT 1858850 E 20150224; RS 53873 B1 20150831; SI 1858850 T1 20150430; TW 200700388 A 20070101; TW 200716548 A 20070501; TW 201302676 A 20130116; TW I414518 B 20131111; TW I500595 B 20150921; US 2006211863 A1 20060921; US 2010036132 A1 20100211; US 2010152460 A1 20100617; US 7629488 B2 20091208; WO 2006098982 A1 20060921; WO 2006099060 A2 20060921; WO 2006099060 A3 20061102; ZA 200708809 B 20090325; ZA 200708810 B 20090128
DOCDB simple family (application)
US 36858806 A 20060306; AR P060100973 A 20060314; AR P060100974 A 20060314; AU 2006223394 A 20060306; AU 2006223482 A 20060306; BR PI0607792 A 20060306; BR PI0607793 A 20060306; CA 2601481 A 20060306; CA 2601674 A 20060306; CN 200680016371 A 20060306; CN 200680016632 A 20060306; CR 9438 A 20071012; CY 151100172 T 20150219; DK 06737611 T 20060306; EA 200701978 A 20060306; EA 200701979 A 20060306; EP 06737413 A 20060306; EP 06737611 A 20060306; ES 06737611 T 20060306; HR P20150417 T 20150414; HU E06737611 A 20060306; IL 18597207 A 20070916; IL 18597407 A 20070916; IL 20940210 A 20101118; JP 2008501912 A 20060306; JP 2008501919 A 20060306; JP 2013147688 A 20130716; KR 20077022664 A 20060306; KR 20077023282 A 20071011; ME P3115 A 20060306; MX 2007011409 A 20060306; MX 2007011412 A 20060306; MY PI20061110 A 20060314; NI 200700237 A 20070913; NO 20075268 A 20071015; NO 20075269 A 20071015; NZ 59057006 A 20060306; PL 06737611 T 20060306; PT 06737611 T 20060306; RS P20150121 A 20060306; SI 200631907 T 20060306; TW 101129655 A 20060314; TW 95108512 A 20060314; TW 95108513 A 20060314; US 2006008240 W 20060306; US 2006008450 W 20060306; US 36856406 A 20060306; US 58064109 A 20091016; US 62597309 A 20091125; ZA 200708809 A 20071012; ZA 200708810 A 20071012