Global Patent Index - EP 1863799 A1

EP 1863799 A1 20071212 - CGRP-ANTAGONISTS, PROCESS FOR THEIR PREPARATION AS WELL AS THEIR USE AS MEDICAMENTS

Title (en)

CGRP-ANTAGONISTS, PROCESS FOR THEIR PREPARATION AS WELL AS THEIR USE AS MEDICAMENTS

Title (de)

CGRP-ANTAGONISTEN, VERFAHREN ZU DEREN HERSTELLUNG SOWIE DEREN VERWENDUNG ALS ARZNEIMITTEL

Title (fr)

ANTAGONISTES CGRP, LEUR PROCÉDÉ DE PRÉPARATION ANSI QUE LEUR UTILISATION COMME MÉDICAMENTS

Publication

EP 1863799 A1 20071212 (DE)

Application

EP 06723538 A 20060318

Priority

  • EP 2006002515 W 20060318
  • EP 2005003094 W 20050323
  • EP 2005004104 W 20050418
  • EP 05021283 A 20050929
  • EP 06723538 A 20060318

Abstract (en)

[origin: WO2006100009A1] The invention relates to CGRP antagonists of general formula (I) in which: R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP> and X are defined as in Claim 1, to their tautomers, isomers, diastereomers, enantiomers, hydrates, mixtures and salts as well as the hydrates of the salts, in particular, their physiologically compatible salts with inorganic or organic acids and bases, and those compounds of general formula (I) in which one or more hydrogen atoms are replaced by deuterium. The invention also relates to medicaments containing these compounds, the use thereof, and to methods for producing them.

IPC 8 full level

C07D 405/12 (2006.01); C07D 405/14 (2006.01); C07D 413/14 (2006.01)

CPC (source: EP KR US)

A61K 31/551 (2013.01 - KR); A61P 1/00 (2017.12 - EP); A61P 1/02 (2017.12 - EP); A61P 1/10 (2017.12 - EP); A61P 3/00 (2017.12 - EP); A61P 3/10 (2017.12 - EP); A61P 5/50 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 11/00 (2017.12 - EP); A61P 11/02 (2017.12 - EP); A61P 11/06 (2017.12 - EP); A61P 17/00 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/06 (2017.12 - EP); A61P 25/36 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 37/08 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 405/12 (2013.01 - EP KR US); C07D 405/14 (2013.01 - EP KR US); C07D 413/14 (2013.01 - EP KR US)

Citation (search report)

See references of WO 2006100009A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

DOCDB simple family (publication)

WO 2006100009 A1 20060928; AU 2006226615 A1 20060928; BR PI0607577 A2 20090915; CA 2600909 A1 20060928; EP 1770091 A1 20070404; EP 1863799 A1 20071212; IL 186090 A0 20080120; JP 2008538209 A 20081016; KR 20070114831 A 20071204; MX 2007011527 A 20071019; US 2006252931 A1 20061109; US 2009186881 A1 20090723; US 2010144716 A1 20100610; US 7528129 B2 20090505; US 7696209 B2 20100413

DOCDB simple family (application)

EP 2006002515 W 20060318; AU 2006226615 A 20060318; BR PI0607577 A 20060318; CA 2600909 A 20060318; EP 05021283 A 20050929; EP 06723538 A 20060318; IL 18609007 A 20070920; JP 2008502299 A 20060318; KR 20077024324 A 20071023; MX 2007011527 A 20060318; US 27717706 A 20060322; US 36317509 A 20090130; US 70789010 A 20100218