EP 1881965 A1 20080130 - 2-AMINO-4-PHENYLQUINAZOLINE DERIVATES AND THEIR USE AS HSP90 MODULATORS
Title (en)
2-AMINO-4-PHENYLQUINAZOLINE DERIVATES AND THEIR USE AS HSP90 MODULATORS
Title (de)
2-AMIN0-4-PHENYLCHINAZOLINDERIVATE UND IHRE VERWENDUNG ALS HSP90 MODULATOREN
Title (fr)
DERIVES DE 2-AMIN0-4-PHENYLCHINAZOLINE ET LEUR UTILISATION COMME MODULATEURS DE HSP90
Publication
Application
Priority
- EP 2006003734 W 20060424
- DE 102005022977 A 20050519
Abstract (en)
[origin: WO2006122631A1] New phenylquinazoline derivatives of the formula (I) in which R<SUP>1</SUP>, R<SUP>2</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP> and R<SUP>5</SUP> are as defined in claim 1 are HSP90 inhibitors and can be used for manufacturing a medicinal product for the treatment of diseases where the inhibition, regulation and/or modulation of HSP90 plays a part.
IPC 8 full level
C07D 239/84 (2006.01); A61K 31/517 (2006.01); C07D 401/12 (2006.01); C07D 403/12 (2006.01)
CPC (source: EP KR US)
A61K 31/517 (2013.01 - KR); A61P 1/00 (2017.12 - EP); A61P 1/04 (2017.12 - EP); A61P 1/16 (2017.12 - EP); A61P 3/00 (2017.12 - EP); A61P 3/10 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 11/00 (2017.12 - EP); A61P 11/06 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 15/00 (2017.12 - EP); A61P 17/00 (2017.12 - EP); A61P 17/02 (2017.12 - EP); A61P 17/06 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 21/00 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/14 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 27/02 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 31/00 (2017.12 - EP); A61P 31/12 (2017.12 - EP); A61P 31/18 (2017.12 - EP); A61P 31/20 (2017.12 - EP); A61P 31/22 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 35/02 (2017.12 - EP); A61P 35/04 (2017.12 - EP); A61P 37/06 (2017.12 - EP); A61P 39/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 239/84 (2013.01 - EP KR US); C07D 401/12 (2013.01 - EP KR US); C07D 403/12 (2013.01 - EP KR US)
Citation (search report)
See references of WO 2006122631A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2006122631 A1 20061123; AR 054047 A1 20070530; AU 2006246744 A1 20061123; AU 2006246744 B2 20111103; BR PI0610134 A2 20100601; CA 2608766 A1 20061123; CN 101180278 A 20080514; CN 101180278 B 20110504; DE 102005022977 A1 20061207; EP 1881965 A1 20080130; HK 1119690 A1 20090313; JP 2008540587 A 20081120; JP 5075117 B2 20121114; KR 20080016651 A 20080221; MX 2007014264 A 20080122; RU 2007146388 A 20090627; RU 2421449 C2 20110620; US 2008214586 A1 20080904; US 7947696 B2 20110524; ZA 200710966 B 20081231
DOCDB simple family (application)
EP 2006003734 W 20060424; AR P060102035 A 20060519; AU 2006246744 A 20060424; BR PI0610134 A 20060424; CA 2608766 A 20060424; CN 200680017419 A 20060424; DE 102005022977 A 20050519; EP 06724519 A 20060424; HK 08111820 A 20081028; JP 2008511580 A 20060424; KR 20077029415 A 20071217; MX 2007014264 A 20060424; RU 2007146388 A 20060424; US 91460406 A 20060424; ZA 200710966 A 20071218