Global Patent Index - EP 1891080 A2

EP 1891080 A2 20080227 - NOVEL PHOSPHORUS-CONTAINING THYROMIMETICS

Title (en)

NOVEL PHOSPHORUS-CONTAINING THYROMIMETICS

Title (de)

NEUE PHOSPHORHALTIGE THYROMIMETIKA

Title (fr)

NOUVELLES SUBSTANCES THYROMIMETIQUES CONTENANT DU PHOSPHORE

Publication

EP 1891080 A2 20080227 (EN)

Application

EP 06760469 A 20060526

Priority

  • US 2006020607 W 20060526
  • US 13777305 A 20050526
  • US 72517005 P 20051006

Abstract (en)

[origin: WO2006128055A2] The present invention relates to compounds of phosphonic acid-containing T3 mimetics and monoesters thereof, stereoisomers, pharmaceutically acceptable salts, co-crystals, and prodrugs thereof and pharmaceutically acceptable salts and co-crystals of the prodrugs, as well as their preparation and uses for preventing and/or treating metabolic diseases such as obesity, NASH, hypercholesterolemia and hyperlipidemia, as well as associated conditions such as atherosclerosis, coronary heart disease, impaired glucose tolerance, metabolic syndrome x and diabetes.

IPC 8 full level

C07F 9/02 (2006.01); C07F 9/30 (2006.01); C07F 9/38 (2006.01); C07F 9/40 (2006.01); C07F 9/44 (2006.01)

CPC (source: EP)

A61P 1/16 (2017.12); A61P 3/04 (2017.12); A61P 3/06 (2017.12); A61P 3/08 (2017.12); A61P 3/10 (2017.12); A61P 5/14 (2017.12); A61P 9/10 (2017.12); A61P 9/12 (2017.12); A61P 43/00 (2017.12); C07F 9/3211 (2013.01); C07F 9/36 (2013.01); C07F 9/3808 (2013.01); C07F 9/3882 (2013.01); C07F 9/4006 (2013.01); C07F 9/4056 (2013.01); C07F 9/4075 (2013.01); C07F 9/4407 (2013.01); C07F 9/4426 (2013.01); C07F 9/4465 (2013.01); C07F 9/65517 (2013.01); C07F 9/657181 (2013.01)

Citation (search report)

See references of WO 2006128055A2

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA HR MK YU

DOCDB simple family (publication)

WO 2006128055 A2 20061130; WO 2006128055 A3 20070524; AU 2006249347 A1 20061130; CA 2606497 A1 20061130; CN 101189248 A 20080528; EP 1891080 A2 20080227; JP 2008545710 A 20081218; MX 2007014493 A 20080207

DOCDB simple family (application)

US 2006020607 W 20060526; AU 2006249347 A 20060526; CA 2606497 A 20060526; CN 200680017732 A 20060526; EP 06760469 A 20060526; JP 2008513783 A 20060526; MX 2007014493 A 20060526