EP 1910341 A2 20080416 - INHIBITORS OF SERINE PROTEASES
Title (en)
INHIBITORS OF SERINE PROTEASES
Title (de)
SERINPROTEASE-HEMMER
Title (fr)
INHIBITEURS DES SERINES PROTEASES
Publication
Application
Priority
- US 2006029988 W 20060801
- US 70477205 P 20050802
Abstract (en)
[origin: WO2007016589A2] This invention relates to compounds of formula (I): or a pharmaceutically acceptable salt or mixtures thereof wherein C* represents a diastereomeric carbon comprising a mixture of R andS isomers wherein the R isomer is greater than 50% of the mixture.
IPC 8 full level
C07D 403/12 (2006.01); A61K 31/501 (2006.01); A61K 38/08 (2019.01); C07K 5/06 (2006.01); C07K 5/10 (2006.01)
CPC (source: EP KR US)
A01N 37/46 (2013.01 - US); A61K 31/497 (2013.01 - US); A61K 31/501 (2013.01 - KR); A61K 38/005 (2013.01 - US); A61K 38/08 (2013.01 - EP US); A61K 45/06 (2013.01 - US); A61P 31/12 (2017.12 - EP); A61P 31/14 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 403/12 (2013.01 - EP KR US); C07K 5/06139 (2013.01 - EP US); C07K 5/1024 (2013.01 - EP US); C07K 7/06 (2013.01 - US); C12N 9/99 (2013.01 - US); A61K 38/00 (2013.01 - EP US)
Citation (search report)
See references of WO 2007016589A2
Citation (third parties)
Third party :
- WO 0218639 A2 20020307 - GEMINI GENOMICS PLC [GB]
- WO 2005042570 A1 20050512 - VERTEX PHARMA [US], et al
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2007016589 A2 20070208; WO 2007016589 A3 20070329; AR 057716 A1 20071212; AU 2006275413 A1 20070208; AU 2006275413 B2 20120719; CA 2617679 A1 20070208; CN 101277950 A 20081001; CN 101277950 B 20130327; EP 1910341 A2 20080416; EP 1910341 B1 20130102; EP 2256113 A1 20101201; EP 2402331 A1 20120104; ES 2401661 T3 20130423; IL 189192 A0 20080605; JP 2009505966 A 20090212; KR 20080033481 A 20080416; MX 2008001528 A 20080404; NO 20081012 L 20080425; NZ 565540 A 20110630; RU 2008108024 A 20090910; RU 2011141559 A 20130420; RU 2441020 C2 20120127; TW 200740813 A 20071101; US 2007105781 A1 20070510; US 2011171175 A1 20110714; US 2013177531 A1 20130711; US 2014056847 A1 20140227; ZA 200801114 B 20081126
DOCDB simple family (application)
US 2006029988 W 20060801; AR P060103374 A 20060802; AU 2006275413 A 20060801; CA 2617679 A 20060801; CN 200680036528 A 20060801; EP 06800633 A 20060801; EP 10171186 A 20060801; EP 11160049 A 20060801; ES 06800633 T 20060801; IL 18919208 A 20080203; JP 2008525128 A 20060801; KR 20087005022 A 20080229; MX 2008001528 A 20060801; NO 20081012 A 20080226; NZ 56554006 A 20060801; RU 2008108024 A 20060801; RU 2011141559 A 20111013; TW 95128293 A 20060802; US 201113051557 A 20110318; US 201313780373 A 20130228; US 201314069638 A 20131101; US 49708706 A 20060801; ZA 200801114 A 20080201