Global Patent Index - EP 1915369 A4

EP 1915369 A4 20100908 - NOVEL SUBSTITUTED 1,2,3-T II AZOLYLMETHYL-BENZOTHIOPHENE OR -INDOLE AND THEIR USE AS LEUKOTIIENE BIOSYNTHESIS INHIBITORS

Title (en)

NOVEL SUBSTITUTED 1,2,3-T II AZOLYLMETHYL-BENZOTHIOPHENE OR -INDOLE AND THEIR USE AS LEUKOTIIENE BIOSYNTHESIS INHIBITORS

Title (de)

NEUE SUBSTITUIERTE 1,2,3-TRIAZOLYLMETHYLBENZOTHIOPHENE ODER ENDOLE UND IHRE VERWENDUNG ALS INHIBITOREN DER LEUKOTRIENBIOSYNTHESE

Title (fr)

NOUVEAU 1,2,3-T II AZOLYLMÉTHYLE-BENZOTHIOPHÈNE SUBSTITUÉS OU -INDOLE ET LEUR UTILISATION EN TANT QU'INHIBITEURS DE BIOSYNTHÈSE LEUKOTIIÈNE

Publication

EP 1915369 A4 20100908 (EN)

Application

EP 06775086 A 20060808

Priority

  • CA 2006001306 W 20060808
  • US 70736205 P 20050811

Abstract (en)

[origin: WO2007016784A1] The instant invention provides compounds of Formula I which are leukotpene biosynthesis inhibitors. Z is a fused (optionally sulfo-oxidized) thiophen ring or a fused pyrrol ring R2-R4 are selected from a variety of substituents Compounds of Formula I are useful as anti-atherosclerotic, anti-asthmatic, anti-allergic, anti¬ inflammatory and cytoprotective agents.

IPC 8 full level

A61K 31/4192 (2006.01); A61P 9/10 (2006.01); A61P 11/06 (2006.01); A61P 29/00 (2006.01); C07D 403/06 (2006.01); C07D 409/06 (2006.01); C07D 409/14 (2006.01)

CPC (source: EP)

A61P 9/10 (2017.12); A61P 11/00 (2017.12); A61P 11/06 (2017.12); A61P 27/16 (2017.12); A61P 29/00 (2017.12); A61P 43/00 (2017.12); C07D 403/06 (2013.01); C07D 409/06 (2013.01); C07D 409/14 (2013.01); C07D 413/14 (2013.01)

Citation (search report)

  • No further relevant documents disclosed
  • See references of WO 2007016784A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

DOCDB simple family (publication)

WO 2007016784 A1 20070215; AU 2006279211 A1 20070215; CA 2618586 A1 20070215; EP 1915369 A1 20080430; EP 1915369 A4 20100908; JP 2009504575 A 20090205

DOCDB simple family (application)

CA 2006001306 W 20060808; AU 2006279211 A 20060808; CA 2618586 A 20060808; EP 06775086 A 20060808; JP 2008525348 A 20060808