Global Patent Index - EP 1919888 A2

EP 1919888 A2 20080514 - METHOD FOR PRODUCING NEBIVOLOL

Title (en)

METHOD FOR PRODUCING NEBIVOLOL

Title (de)

VERFAHREN ZUR HERSTELLUNG NEBIVOLOL

Title (fr)

PROCEDE DE PRODUCTION DE NEBIVOLOL

Publication

EP 1919888 A2 20080514 (DE)

Application

EP 06760790 A 20060717

Priority

  • AT 2006000303 W 20060717
  • AT 12142005 A 20050719

Abstract (en)

[origin: WO2007009143A2] The invention relates to a method for producing the racemic active ingredient Nebivolol, according to which diastereomer cyanhydrins are produced and separated, and the separated diastereomers are coupled together following a transformation, preferably a partial or full reduction of the cyano group or a Pinner saponification.

IPC 8 full level

C07D 311/58 (2006.01); C07F 7/18 (2006.01)

CPC (source: EP KR US)

C07D 311/58 (2013.01 - EP US); C07D 407/12 (2013.01 - KR)

Citation (search report)

See references of WO 2007009143A2

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA HR MK RS

DOCDB simple family (publication)

WO 2007009143 A2 20070125; WO 2007009143 A3 20070405; AT 502220 A1 20070215; AU 2006272420 A1 20070125; BR PI0613610 A2 20110118; CA 2615832 A1 20070125; CN 101243062 A 20080813; EA 200800364 A1 20080630; EP 1919888 A2 20080514; IL 188777 A0 20080807; JP 2009502750 A 20090129; KR 20080027368 A 20080326; MX 2008000747 A 20080414; NO 20080823 L 20080402; US 2008221340 A1 20080911; ZA 200800963 B 20090826

DOCDB simple family (application)

AT 2006000303 W 20060717; AT 12142005 A 20050719; AU 2006272420 A 20060717; BR PI0613610 A 20060717; CA 2615832 A 20060717; CN 200680029362 A 20060717; EA 200800364 A 20060717; EP 06760790 A 20060717; IL 18877708 A 20080115; JP 2008521739 A 20060717; KR 20087001837 A 20080123; MX 2008000747 A 20060717; NO 20080823 A 20080215; US 99637006 A 20060717; ZA 200800963 A 20060717