Global Patent Index - EP 1937640 A2

EP 1937640 A2 20080702 - 1,2,3,5-TETRAHYDRO-CYCLOPENTAL[C]QUINOLIN-4-ONE DERIVATIVES AS RXR AGONISTS FOR THE TREATMENT OF DYSLIPIDEMIA, HYPERCHOLESTEROLEMIA AND DIABETES

Title (en)

1,2,3,5-TETRAHYDRO-CYCLOPENTAL[C]QUINOLIN-4-ONE DERIVATIVES AS RXR AGONISTS FOR THE TREATMENT OF DYSLIPIDEMIA, HYPERCHOLESTEROLEMIA AND DIABETES

Title (de)

1,2,3,5-TETRAHYDROCYCLOPENTAL[C]CHINOLIN-4-ONDERIVATE ALS RXR-AGONISTEN ZUR BEHANDLUNG VON DYSLIPIDÄMIE, HYPERCHOLESTERINÄMIE UND DIABETES

Title (fr)

DERIVES DE 1,2,3,5-TETRAHYDRO-CYCLOPENTAL[C]QUINOLIN-4-ONE UTILISES EN TANT QU'AGONISTES DU RECEPTEUR RXR POUR LE TRAITEMENT DE LA DYSLIPIDEMIE, DE L'HYPERCHOLESTEROLEMIE ET DU DIABETE

Publication

EP 1937640 A2 20080702 (EN)

Application

EP 06815371 A 20060925

Priority

  • US 2006037321 W 20060925
  • US 72250705 P 20050930

Abstract (en)

[origin: WO2007041076A2] The present invention relates to compounds of Formula (I), methods for preparing these compounds, compositions, intermediates and derivatives thereof and for treating RXR mediated disorders. More particularly, the compounds of the present invention are RXR agonists useful for treating RXR mediated disorders.

IPC 8 full level

C07D 215/22 (2006.01); A61K 31/473 (2006.01); A61P 3/06 (2006.01); A61P 3/10 (2006.01); A61P 9/10 (2006.01); A61P 29/00 (2006.01)

CPC (source: EP)

A61P 1/04 (2017.12); A61P 3/02 (2017.12); A61P 3/04 (2017.12); A61P 3/06 (2017.12); A61P 3/10 (2017.12); A61P 5/50 (2017.12); A61P 7/02 (2017.12); A61P 9/00 (2017.12); A61P 9/10 (2017.12); A61P 9/12 (2017.12); A61P 13/12 (2017.12); A61P 15/00 (2017.12); A61P 25/00 (2017.12); A61P 27/02 (2017.12); A61P 27/12 (2017.12); A61P 29/00 (2017.12); A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07D 215/233 (2013.01)

Citation (search report)

See references of WO 2007041076A2

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR

DOCDB simple family (publication)

WO 2007041076 A2 20070412; WO 2007041076 A3 20070607; CA 2624345 A1 20070412; CN 101316822 A 20081203; EP 1937640 A2 20080702; JP 2009510071 A 20090312

DOCDB simple family (application)

US 2006037321 W 20060925; CA 2624345 A 20060925; CN 200680044332 A 20060925; EP 06815371 A 20060925; JP 2008533489 A 20060925