EP 1939204 B3 20220824 - FUSED HETEROCYCLIC DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF
Title (en)
FUSED HETEROCYCLIC DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE SAME, AND MEDICINAL USE THEREOF
Title (de)
KONDENSIERTES HETEROCYCLISCHES DERIVAT, DIESES ENTHALTENDE MEDIZINISCHE ZUSAMMENSETZUNG UND DEREN MEDIZINISCHE VERWENDUNG
Title (fr)
DÉRIVÉ HÉTÉROCYCLIQUE À CYCLES JOINTS, PRÉPARATION THÉRAPEUTIQUE CONTENANT LEDIT DÉRIVÉ, ET EMPLOI THÉRAPEUTIQUE DUDIT DÉRIVÉ
Publication
Application
Priority
- JP 2006320681 W 20061017
- JP 2005304395 A 20051019
- JP 2006147019 A 20060526
Abstract (en)
[origin: EP1939204A1] The present invention provides a compound useful as an agent for the prevention or treatment of a sex hormone-dependent disease or the like. That is, the present invention provides a fused heterocyclic derivative represented by the following general formula (I), a pharmaceutical composition containing the same, a medicinal use thereof and the like. In the formula (I), ring A represents 5-membered cyclic unsaturated hydrocarbon or 5-membered heteroaryl; R A represents halogen, alkyl, alkenyl, alkynyl, carboxy, alkoxy, carbamoyl, alkylcarbamoyl or the like; ring B represents aryl or heteroaryl; R B represents halogen, alkyl, carboxy, alkoxy, carbamoyl, alkylcarbamoyl or the like; E 1 and E 2 represent an oxygen atom or the like; U represents a single bond or alkylene; X represents a group represented by Y, -SO 2 -Y, -O-(alkylene)-Y, -O-Z in which Y represents Z, amino or the like; Z represents cycloalkyl, heterocycloalkyl, aryl, heteroaryl or the like; or the like.
IPC 8 full level
C07D 487/04 (2006.01); A61K 31/519 (2006.01); A61K 31/55 (2006.01); A61K 45/00 (2006.01); A61P 13/08 (2006.01); A61P 15/00 (2006.01); A61P 15/18 (2006.01); A61P 17/02 (2006.01); A61P 17/10 (2006.01); A61P 17/14 (2006.01); A61P 19/00 (2006.01); A61P 25/20 (2006.01); A61P 25/28 (2006.01); A61P 35/00 (2006.01); A61P 43/00 (2006.01); C07D 495/04 (2006.01)
CPC (source: EP KR NO US)
A61K 31/519 (2013.01 - KR NO); A61K 31/55 (2013.01 - KR); A61P 1/00 (2018.01 - EP); A61P 5/04 (2018.01 - EP); A61P 5/24 (2018.01 - EP); A61P 5/28 (2018.01 - EP); A61P 5/32 (2018.01 - EP); A61P 13/00 (2018.01 - EP); A61P 13/08 (2018.01 - EP); A61P 15/00 (2018.01 - EP NO); A61P 15/08 (2018.01 - EP); A61P 15/18 (2018.01 - EP); A61P 17/00 (2018.01 - EP); A61P 17/02 (2018.01 - EP); A61P 17/10 (2018.01 - EP); A61P 17/14 (2018.01 - EP); A61P 19/00 (2018.01 - EP); A61P 25/00 (2018.01 - EP); A61P 25/20 (2018.01 - EP); A61P 25/28 (2018.01 - EP); A61P 35/00 (2018.01 - EP NO); A61P 43/00 (2018.01 - EP NO); C07D 487/04 (2013.01 - KR); C07D 495/04 (2013.01 - EP NO US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
EP 1939204 A1 20080702; EP 1939204 A4 20100901; EP 1939204 B1 20130102; EP 1939204 B3 20220824; AU 2006305271 A1 20070426; AU 2006305271 B2 20111117; BR PI0617436 A2 20110726; BR PI0617436 B1 20210406; BR PI0617436 B8 20210525; CA 2624492 A1 20070426; CA 2624492 C 20140218; CY 1113898 T1 20160727; DK 1939204 T3 20130311; DK 1939204 T6 20220905; ES 2398917 T3 20130322; ES 2398917 T7 20221026; HK 1125110 A1 20090731; IL 190754 A0 20081103; IL 190754 A 20121031; JP 2012102140 A 20120531; JP 4955566 B2 20120620; JP 5319797 B2 20131016; JP WO2007046392 A1 20090423; KR 101384132 B1 20140410; KR 20080063827 A 20080707; NL 301202 I1 20221109; NL 301202 I2 20230124; NO 20082249 L 20080718; NO 343185 B1 20181126; NZ 567300 A 20101126; PL 1939204 T3 20130628; PL 1939204 T6 20240325; PT 1939204 E 20130314; RU 2008119462 A 20091127; RU 2418803 C2 20110520; SI 1939204 T1 20130531; TW 200732309 A 20070901; TW I400074 B 20130701; US 2009325900 A1 20091231; US 9040693 B2 20150526; WO 2007046392 A1 20070426
DOCDB simple family (application)
EP 06811925 A 20061017; AU 2006305271 A 20061017; BR PI0617436 A 20061017; CA 2624492 A 20061017; CY 131100276 T 20130402; DK 06811925 T 20061017; ES 06811925 T 20061017; HK 09103380 A 20090409; IL 19075408 A 20080409; JP 2006320681 W 20061017; JP 2007540993 A 20061017; JP 2012008680 A 20120119; KR 20087010997 A 20061017; NL 301202 C 20221101; NO 20082249 A 20080519; NZ 56730006 A 20061017; PL 06811925 T 20061017; PT 06811925 T 20061017; RU 2008119462 A 20061017; SI 200631557 T 20061017; TW 95138520 A 20061019; US 8967406 A 20061017