EP 1979319 A1 20081015 - NOVEL DUAL NK2/NK3-ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND PROCESSES FOR THEIR PREPARATIONS
Title (en)
NOVEL DUAL NK2/NK3-ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND PROCESSES FOR THEIR PREPARATIONS
Title (de)
NEUE DUALE NK2/NK3-ANTAGONISTEN, PHARMAZEUTISCHE ZUSAMMENSETZUNGEN, DIE SIE ENTHALTEN, UND VERFAHREN ZU IHRER HERSTELLUNG
Title (fr)
NOUVEAUX ANTAGONISTES DOUBLES DE NK2/NK3, COMPOSITIONS PHARMACEUTIQUES LES COMPRENANT ET LEURS PROCEDES DE PREPARATION
Publication
Application
Priority
- EP 2007050964 W 20070201
- EP 06101139 A 20060201
- EP 07704286 A 20070201
Abstract (en)
[origin: WO2007088181A1] The present invention relates to novel dual NK2/NK3-antagonists of formula (I) wherein the meaning of X and R1 to R5 is defined in the claims and in the description and also to pharmaceutical compositions comprising these compounds. Furthermore, the invention relates to processes for the preparation of the novel dual NK2/NK3-antagonists and to their uses.
IPC 8 full level
C07D 211/66 (2006.01); A61K 31/44 (2006.01); A61K 31/443 (2006.01); A61K 31/4433 (2006.01); A61K 31/4439 (2006.01); A61K 31/444 (2006.01); A61K 31/445 (2006.01); C07D 211/58 (2006.01); C07D 211/62 (2006.01); C07D 295/14 (2006.01); C07D 401/04 (2006.01); C07D 401/12 (2006.01); C07D 405/12 (2006.01); C07D 409/12 (2006.01); C07D 413/12 (2006.01)
CPC (source: EP)
A61P 1/04 (2017.12); A61P 9/00 (2017.12); A61P 9/12 (2017.12); A61P 11/00 (2017.12); A61P 11/02 (2017.12); A61P 11/06 (2017.12); A61P 13/02 (2017.12); A61P 17/00 (2017.12); A61P 17/06 (2017.12); A61P 19/02 (2017.12); A61P 25/00 (2017.12); A61P 25/04 (2017.12); A61P 25/06 (2017.12); A61P 25/18 (2017.12); A61P 25/22 (2017.12); A61P 25/24 (2017.12); A61P 25/28 (2017.12); A61P 35/00 (2017.12); A61P 43/00 (2017.12); C07D 211/58 (2013.01); C07D 211/62 (2013.01); C07D 211/66 (2013.01); C07D 295/155 (2013.01); C07D 401/04 (2013.01); C07D 401/12 (2013.01); C07D 405/12 (2013.01); C07D 409/12 (2013.01); C07D 413/12 (2013.01)
Citation (search report)
See references of WO 2007088181A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2007088181 A1 20070809; AU 2007211475 A1 20070809; CA 2641817 A1 20070809; CN 101374811 A 20090225; EP 1979319 A1 20081015; JP 2009525308 A 20090709; RU 2008135123 A 20100310
DOCDB simple family (application)
EP 2007050964 W 20070201; AU 2007211475 A 20070201; CA 2641817 A 20070201; CN 200780003129 A 20070201; EP 07704286 A 20070201; JP 2008552803 A 20070201; RU 2008135123 A 20070201