EP 1979333 A1 20081015 - PROCESS FOR PREPARING IODINATED AZOLES
Title (en)
PROCESS FOR PREPARING IODINATED AZOLES
Title (de)
VERFAHREN ZUR HERSTELLUNG VON IODIERTEN AZOLEN
Title (fr)
PROCEDE DE FABRICATION D'AZOLES IODES
Publication
Application
Priority
- EP 2007000236 W 20070112
- DE 102006003444 A 20060125
Abstract (en)
[origin: DE102006003444A1] Method for iodinating substituted azole compound (I) or its salts and acid addition compounds by converting substituted 1H-triazoles (II) or its salts and acid addition compounds with oxidizing agent and elementary iodine and/or at least one iodine compound in presence of a solvent or its mixture at 0-200[deg]C. Method for iodinating substituted azole compound of formula (I) or its salts and acid addition compounds by converting substituted 1H-triazoles compound of formula (II) or its salts and acid addition compounds with at least one oxidizing agent and elementary iodine and/or at least one iodine compound in presence of a solvent or its mixture at 0-200[deg]C. A : N, CH or CR 3; B 1>N, CH, CR 4or Cl; R 1>alkenyl, alkynyl, (cyclo)alkyl, phenyl (all optionally substituted) or H; R 2>I; and R 3>, R 4>alkenyl, alkynyl, (cyclo)alkyl, phenyl or phenyl ethyl (all optionally substituted). . Provided that at least one of A and B 1>is N. [Image] ACTIVITY : Antibacterial. MECHANISM OF ACTION : None given.
IPC 8 full level
C07D 257/04 (2006.01); C07D 249/10 (2006.01)
CPC (source: EP US)
C07D 249/10 (2013.01 - EP US); C07D 257/04 (2013.01 - EP US)
Citation (search report)
See references of WO 2007085349A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
DE 102006003444 A1 20070726; EP 1979333 A1 20081015; JP 2009524610 A 20090702; US 2011015403 A1 20110120; WO 2007085349 A1 20070802
DOCDB simple family (application)
DE 102006003444 A 20060125; EP 07702709 A 20070112; EP 2007000236 W 20070112; JP 2008551690 A 20070112; US 22313407 A 20070112