EP 2010513 A2 20090107 - NOVEL CRYSTALLINE COMPOUNDS
Title (en)
NOVEL CRYSTALLINE COMPOUNDS
Title (de)
NEUE KRISTALLINE VERBINDUNGEN
Title (fr)
NOUVEAUX COMPOSÉS CRISTALLINS
Publication
Application
Priority
- EP 2007053488 W 20070411
- DE 102006017827 A 20060413
Abstract (en)
[origin: WO2007118819A2] The invention relates to the novel crystalline compounds A of general formula I, wherein A<SUP>1</SUP>, A<SUP>2</SUP>, A<SUP>3</SUP>, X, Y<SUP>1</SUP>, Y<SUP>2</SUP>, and Y<SUP>3</SUP> are defined as indicated in claim 1, and which are provided in the form of the physiologically acceptable salts thereof with acids, said acids being selected among group B comprising hydrochloric acid, hydrobromic acid, sulfuric acid, phosphoric acid, benzenesulfonic acid, p-toluenesulfonic acid, maleic acid, succinic acid, fumaric acid, D-(-)-tartaric acid, L-(+)-tartaric acid, naphthalene-2-sulfonic acid, and naphthalene-1,5-disulfonic acid, as well as the polymorphs, the respective solvates and hydrates.
IPC 8 full level
C07D 401/04 (2006.01)
CPC (source: EP KR US)
A61K 31/551 (2013.01 - KR); A61P 1/12 (2017.12 - EP); A61P 3/10 (2017.12 - EP); A61P 5/30 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 11/00 (2017.12 - EP); A61P 11/02 (2017.12 - EP); A61P 11/06 (2017.12 - EP); A61P 15/08 (2017.12 - EP); A61P 17/00 (2017.12 - EP); A61P 17/02 (2017.12 - EP); A61P 17/04 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 25/04 (2017.12 - EP); A61P 25/06 (2017.12 - EP); A61P 25/36 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 37/08 (2017.12 - EP); C07D 401/04 (2013.01 - EP KR US); C07D 401/14 (2013.01 - EP KR US)
Citation (search report)
See references of WO 2007118819A2
Citation (examination)
- STAHL; WERMUTH: "Handbook of Pharmaceutical Salts - Properties, Selection, and Use", 2002, WILEY-VCH, Weinheim, ISBN: 3906390268, pages: 191-193, 211-214, 308
- HILFIKER: "Polymorphism in the Pharmaceutical Industry", 2006, WILEY-VCH, Weinheim, ISBN: 3527311460, pages: 274
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA HR MK RS
DOCDB simple family (publication)
DE 102006017827 A1 20071018; AR 060442 A1 20080618; AU 2007239505 A1 20071025; BR PI0710151 A2 20110802; CA 2648140 A1 20071025; CN 101421263 A 20090429; CO 6140057 A2 20100319; EA 200802049 A1 20090428; EC SP088737 A 20081031; EP 2010513 A2 20090107; JP 2009533387 A 20090917; KR 20090007428 A 20090116; MX 2008013158 A 20081022; NO 20083709 L 20081031; PE 20080735 A1 20080725; TW 200808767 A 20080216; US 2008086003 A1 20080410; US 7638625 B2 20091229; UY 30280 A1 20071130; WO 2007118819 A2 20071025; WO 2007118819 A3 20080529; ZA 200806859 B 20090826
DOCDB simple family (application)
DE 102006017827 A 20060413; AR P070101573 A 20070413; AU 2007239505 A 20070411; BR PI0710151 A 20070411; CA 2648140 A 20070411; CN 200780012808 A 20070411; CO 08108825 A 20081010; EA 200802049 A 20070411; EC SP088737 A 20080915; EP 07727956 A 20070411; EP 2007053488 W 20070411; JP 2009504732 A 20070411; KR 20087027714 A 20081112; MX 2008013158 A 20070411; NO 20083709 A 20080828; PE 2007000446 A 20070411; TW 96112795 A 20070412; US 73452007 A 20070412; UY 30280 A 20070412; ZA 200806859 A 20080808