EP 2089381 A1 20090819 - INDOLES WHICH ACT AS VIA RECEPTOR ANTAGONISTS
Title (en)
INDOLES WHICH ACT AS VIA RECEPTOR ANTAGONISTS
Title (de)
ALS VIA-REZEPTOR-ANTAGONISTEN VERWENDBARE INDOLE
Title (fr)
INDOLES AGISSANT COMME DES ANTAGONISTES DU RÉCEPTEUR V1A
Publication
Application
Priority
- EP 2007062984 W 20071129
- EP 06125663 A 20061208
- EP 07847501 A 20071129
Abstract (en)
[origin: WO2008068184A1] The present invention is concerned with novel indol-2-yl-carbonyl-piperidin- benzoimidazolon and indol-2-yl-carbonyl-piperidin-benzoxazolon derivatives as V1a receptor antagonists, their manufacture, pharmaceutical compositions containing them and their use as medicaments. The active compounds of the present invention are useful in the prevention and/or treatment of anxiety and depressive disorders and other diseases. Present invention comprises compounds of the general formula (I) wherein R<SUP>1</SUP> to R<SUP>11</SUP>, X and Y are as defined in the specification.
IPC 8 full level
C07D 401/14 (2006.01); A61K 31/4427 (2006.01); A61P 25/22 (2006.01); A61P 25/24 (2006.01); C07D 491/04 (2006.01)
CPC (source: EP KR US)
A61K 31/4427 (2013.01 - KR); A61P 1/16 (2017.12 - EP); A61P 5/02 (2017.12 - EP); A61P 5/24 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/02 (2017.12 - EP); A61P 9/04 (2017.12 - EP); A61P 9/12 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 15/00 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/22 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 401/14 (2013.01 - EP KR US); C07D 491/04 (2013.01 - EP KR US)
Citation (search report)
See references of WO 2008068184A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2008068184 A1 20080612; AR 064137 A1 20090318; AT E472544 T1 20100715; AU 2007328994 A1 20080612; AU 2007328994 B2 20120308; BR PI0720441 A2 20140107; CA 2671324 A1 20080612; CL 2007003503 A1 20080704; CN 101541786 A 20090923; DE 602007007512 D1 20100812; EP 2089381 A1 20090819; EP 2089381 B1 20100630; ES 2345132 T3 20100915; IL 198683 A0 20100217; JP 2010511660 A 20100415; KR 101050558 B1 20110719; KR 20090078368 A 20090717; MX 2009005541 A 20090605; NO 20091832 L 20090707; PE 20081380 A1 20080918; RU 2009120443 A 20110120; TW 200829570 A 20080716; US 2008139548 A1 20080612; US 2008139617 A1 20080612; US 2008139618 A1 20080612; US 2008269290 A1 20081030; US 7799923 B2 20100921; US 8071622 B2 20111206; ZA 200903499 B 20100331
DOCDB simple family (application)
EP 2007062984 W 20071129; AR P070105428 A 20071205; AT 07847501 T 20071129; AU 2007328994 A 20071129; BR PI0720441 A 20071129; CA 2671324 A 20071129; CL 2007003503 A 20071205; CN 200780042134 A 20071129; DE 602007007512 T 20071129; EP 07847501 A 20071129; ES 07847501 T 20071129; IL 19868309 A 20090511; JP 2009539706 A 20071129; KR 20097011629 A 20071129; MX 2009005541 A 20071129; NO 20091832 A 20090511; PE 2007001745 A 20071207; RU 2009120443 A 20071129; TW 96146544 A 20071206; US 94714607 A 20071129; US 94719507 A 20071129; US 94726607 A 20071129; US 99837107 A 20071129; ZA 200903499 A 20090520