Global Patent Index - EP 2097410 A1

EP 2097410 A1 20090909 - HETEROARYL-PYRAZOLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS

Title (en)

HETEROARYL-PYRAZOLE DERIVATIVES AS CANNABINOID CB1 RECEPTOR ANTAGONISTS

Title (de)

HETEROARYLPYRAZOLDERIVATE ALS ANTAGONISTEN DES CANNABINOID-CB1-REZEPTORS

Title (fr)

DÉRIVÉS D'HÉTÉROARYL-PYRAZOLE UTILISÉS EN TANT QU'ANTAGONISTES DU RÉCEPTEUR CB1 DES CANNABINOÏDES

Publication

EP 2097410 A1 20090909 (EN)

Application

EP 07833072 A 20070928

Priority

  • KR 2007004754 W 20070928
  • US 54126906 A 20060929
  • KR 20060132606 A 20061222

Abstract (en)

[origin: WO2008039023A1] A heteroaryl-pyrazole compound of formula (I) or a pharmaceutically acceptable salt thereof is effective as a cannabinoid CB1 receptor inverse agonist or antagonist, which is useful for preventing or treating obesity and obesity-related metabolic disorders. The present invention also provides a method for preparing the inventive heteroaryl-pyrasole compounds or a pharmaceutically acceptable salt thereof, a pharmaceutical composition containing same, and a method for preventing or treating obesity and obesity-related metabolic disorders.

IPC 8 full level

A61K 31/415 (2006.01); A61K 31/4155 (2006.01); A61P 3/04 (2006.01); A61P 29/00 (2006.01); C07D 401/14 (2006.01); C07D 403/04 (2006.01); C07D 403/14 (2006.01); C07D 405/14 (2006.01); C07D 409/14 (2006.01); C07D 413/04 (2006.01); C07D 413/14 (2006.01); C07D 417/04 (2006.01); C07D 417/14 (2006.01); C07D 419/04 (2006.01)

CPC (source: EP KR)

A61P 3/04 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 401/14 (2013.01 - EP); C07D 403/04 (2013.01 - EP KR); C07D 403/14 (2013.01 - EP); C07D 405/14 (2013.01 - EP); C07D 409/14 (2013.01 - EP); C07D 413/04 (2013.01 - EP KR); C07D 413/14 (2013.01 - EP); C07D 417/04 (2013.01 - EP KR); C07D 417/14 (2013.01 - EP)

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA HR MK RS

DOCDB simple family (publication)

WO 2008039023 A1 20080403; CN 101528740 A 20090909; CN 101528740 B 20120919; EP 2097410 A1 20090909; EP 2097410 A4 20091125; JP 2010504961 A 20100218; JP 5269795 B2 20130821; KR 101100028 B1 20111229; KR 20090061076 A 20090615

DOCDB simple family (application)

KR 2007004754 W 20070928; CN 200780036330 A 20070928; EP 07833072 A 20070928; JP 2009530273 A 20070928; KR 20097008743 A 20070928