Global Patent Index - EP 2114954 B1

EP 2114954 B1 20130213 - BICYCLIC ARYL AND BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS

Title (en)

BICYCLIC ARYL AND BICYCLIC HETEROARYL SUBSTITUTED TRIAZOLES USEFUL AS AXL INHIBITORS

Title (de)

DURCH BICYCLISCHES ARYL BZW. BICYCLISCHES HETEROARYL SUBSTITUIERTE TRIAZOLE, DIE SICH ALS AXL-INIHIBITOREN EIGNEN

Title (fr)

TRIAZOLES À SUBSTITUTION ARYLE BICYCLIQUES ET HÉTÉROARYLE BICYCLIQUES UTILES EN TANT QU'INHIBITEURS AXL

Publication

EP 2114954 B1 20130213 (EN)

Application

EP 07866121 A 20071228

Priority

  • US 2007089152 W 20071228
  • US 88276906 P 20061229
  • US 97534607 P 20070926

Abstract (en)

[origin: WO2008083353A1] Bicyclic aryl substituted triazoles or heteroaryl substituted triazoles and pharmaceutical compositions containing the compounds are disclosed as being useful in inhibiting the activity of the receptor protein tyrosine kinase Axl. Methods of using the compounds in treating diseases or conditions associated with Axl activity are also disclosed.

IPC 8 full level

A61K 31/4196 (2006.01); A61P 19/00 (2006.01); C07D 249/14 (2006.01); C07D 401/04 (2006.01); C07D 401/14 (2006.01); C07D 403/04 (2006.01); C07D 403/14 (2006.01); C07D 409/14 (2006.01); C07D 417/14 (2006.01); C07D 495/04 (2006.01)

CPC (source: EP US)

A61K 31/395 (2013.01 - EP US); A61K 31/519 (2013.01 - EP US); A61P 9/00 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 17/06 (2017.12 - EP); A61P 19/00 (2017.12 - EP); A61P 19/10 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 35/02 (2017.12 - EP); C07D 401/14 (2013.01 - EP US); C07D 403/04 (2013.01 - EP US); C07D 403/14 (2013.01 - EP US); C07D 417/14 (2013.01 - EP US); C07D 495/04 (2013.01 - EP US)

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR

DOCDB simple family (publication)

WO 2008083353 A1 20080710; CA 2710043 A1 20080708; CA 2710043 C 20160209; EP 2114954 A1 20091111; EP 2114954 B1 20130213; ES 2406930 T3 20130610; US 2008188454 A1 20080807; US 2011071133 A1 20110324; US 2013281468 A1 20131024; US 7872000 B2 20110118; US 8492373 B2 20130723; US 8809347 B2 20140819

DOCDB simple family (application)

US 2007089152 W 20071228; CA 2710043 A 20071228; EP 07866121 A 20071228; ES 07866121 T 20071228; US 201313918697 A 20130614; US 95782210 A 20101201; US 96658507 A 20071228