EP 2120931 A1 20091125 - PYRAZOLE DERIVATIVES AS MODULATORS OF CANNABINOID RECEPTOR
Title (en)
PYRAZOLE DERIVATIVES AS MODULATORS OF CANNABINOID RECEPTOR
Title (de)
PYRAZOL-DERIVATE ALS MODULATOREN DES CANNABINOID-REZEPTORS
Title (fr)
DÉRIVÉS DE PYRAZOLE UTILISÉS EN TANT QUE MODULATEURS DU RÉCEPTEUR CANNABINOÏDE
Publication
Application
Priority
- GB 2007004703 W 20071210
- GB 0625196 A 20061218
Abstract (en)
[origin: WO2008074982A1] Compounds of formula (I) suppress the normal signalling activity of CB1 receptors, and are useful in the treatment of, for example obesity or overweight formula (I): wherein A<SUB>1</SUB>, A<SUB>2</SUB>, A<SUB>5</SUB>, A<SUB>6</SUB>, R<SUB>1</SUB>, R<SUB>2</SUB>, R<SUB>3</SUB>, and X are as defined in the claims.
IPC 8 full level
A61K 31/4155 (2006.01); A61P 3/04 (2006.01); C07D 401/04 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 403/04 (2006.01)
CPC (source: EP)
A61P 3/04 (2017.12); C07D 401/04 (2013.01); C07D 401/12 (2013.01); C07D 401/14 (2013.01); C07D 403/04 (2013.01)
Citation (search report)
See references of WO 2008074982A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HU IE IS IT LI LT LU LV MC MT NL PL PT RO SE SI SK TR
DOCDB simple family (publication)
WO 2008074982 A1 20080626; CA 2673358 A1 20080626; EP 2120931 A1 20091125; GB 0625196 D0 20070124
DOCDB simple family (application)
GB 2007004703 W 20071210; CA 2673358 A 20071210; EP 07848451 A 20071210; GB 0625196 A 20061218