Global Patent Index - EP 2130540 A1

EP 2130540 A1 20091209 - Pharmaceutical compositions containing a crystalline form of posaconazole

Title (en)

Pharmaceutical compositions containing a crystalline form of posaconazole

Title (de)

Pharmazeutische Zusammensetzungen mit einer kristallinen Form von Posaconazol

Title (fr)

Compositions pharmaceutiques contenant une forme cristalline du posaconazole

Publication

EP 2130540 A1 20091209 (EN)

Application

EP 08157435 A 20080602

Priority

EP 08157435 A 20080602

Abstract (en)

The present invention relates to a pharmaceutical composition comprising crystalline form Y of posaconazole. The pharmaceutical composition can be used to treat or prevent fungal infections.

IPC 8 full level

A61K 31/496 (2006.01); A61P 31/10 (2006.01)

CPC (source: EP US)

A61K 31/496 (2013.01 - EP US); A61P 31/00 (2017.12 - EP); A61P 31/10 (2017.12 - EP); Y10T 428/2982 (2015.01 - US)

Citation (applicant)

Citation (search report)

  • [XD] WO 9918097 A1 19990415 - SCHERING CORP [US], et al
  • [XD] WO 9517407 A1 19950629 - SCHERING CORP [US], et al
  • [X] US 5625064 A 19970429 - ANDREWS DAVID R [US], et al
  • [XD] WO 2005117831 A1 20051215 - SCHERING CORP [US], et al
  • [XD] US 5834472 A 19981110 - SANGEKAR SURENDRA A [US], et al
  • [XD] US 5972381 A 19991026 - SANGEKAR SURENDRA A [US], et al
  • [XD] WO 02080678 A1 20021017 - SCHERING CORP [US], et al
  • [X] WO 2007143390 A1 20071213 - ELAN PHARMA INT LTD [IE], et al
  • [X] WO 2006130177 A1 20061207 - SCHERING CORP [US], et al
  • [X] BENNETT ET AL: "Hydroxylated analogues of the orally active broad spectrum antifungal, Sch 51048 (1), and the discovery of posaconazole [Sch 56592; 2 or (S,S)-5]", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, ELSEVIER SCIENCE, GB, vol. 16, no. 1, 1 January 2006 (2006-01-01), pages 186 - 190, XP005168889, ISSN: 0960-894X
  • [X] SAKSENA A K ET AL: "Stereoselective Grignard additions to N-formyl hydrazone: a concise synthesis of Noxafil<R> side chain and a synthesis of Noxafil<R>", TETRAHEDRON LETTERS, ELSEVIER, AMSTERDAM, vol. 45, no. 44, 25 October 2004 (2004-10-25), pages 8249 - 8251, XP004591093, ISSN: 0040-4039
  • [X] ZHOU, WEICHENG ET AL: "Progress in syntheses of azole antifungal agents", ZHONGGUO YIYAO GONGYE ZAZHI , 37(2), 125-133 CODEN: ZYGZEA; ISSN: 1001-8255, 2006, XP009106603
  • [X] SAKSENA, A. K. ET AL: "Advances in the chemistry of novel broad-spectrum orally active azole antifungals: recent studies leading to the discovery of SCH 56592", SPECIAL PUBLICATION - ROYAL SOCIETY OF CHEMISTRY , 198(ANTI-INFECTIVES), 180-199 CODEN: SROCDO; ISSN: 0260-6291, 1997, XP009106585

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA MK RS

DOCDB simple family (publication)

EP 2130540 A1 20091209; CA 2726704 A1 20091210; CA 2726704 C 20161025; CN 102046172 A 20110504; CN 102046172 B 20130619; DK 2318004 T3 20130708; EP 2318004 A2 20110511; EP 2318004 B1 20130410; ES 2416485 T3 20130801; SI 2318004 T1 20130731; US 2011105525 A1 20110505; US 8563555 B2 20131022; WO 2009147075 A2 20091210; WO 2009147075 A3 20100128

DOCDB simple family (application)

EP 08157435 A 20080602; CA 2726704 A 20090528; CN 200980119683 A 20090528; DK 09757457 T 20090528; EP 09757457 A 20090528; EP 2009056574 W 20090528; ES 09757457 T 20090528; SI 200930637 T 20090528; US 99329709 A 20090528