EP 2132182 A2 20091216 - AMORPHOUS SOLID COMPOSITION CONTAINING A PYRAZOLE-3-CARBOXAMIDE IN AMORPHOUS FORM AND STABILISING CARRIERS
Title (en)
AMORPHOUS SOLID COMPOSITION CONTAINING A PYRAZOLE-3-CARBOXAMIDE IN AMORPHOUS FORM AND STABILISING CARRIERS
Title (de)
AMORPHE FESTE ZUSAMMENSETZUNG MIT EINEM PYRAZOL-3-CARBOXAMID IN AMORPHER FORM UND STABILISIERENDEN TRÄGERSTOFFEN
Title (fr)
SOLUTION SOLIDE AMORPHE CONTENANT UN DERIVE DE PYRAZOLE-3-CARBOXAMIDE SOUS FORME AMORPHE ET DES EXCIPIENTS STABILISATEURS
Publication
Application
Priority
- FR 2008000216 W 20080220
- FR 0701377 A 20070223
Abstract (en)
[origin: FR2913018A1] Pyrazol-3-carboxamide derivative (I) in amorphous form comprising surinabant and rimonabant form, is new. Independent claims are included for: (1) amorphous solid solution comprising (I) or its salts and/or solvate, with more excipient stabilizers themselves in amorphous form; (2) a preparation of the amorphous solid solution comprising dissolving (I) in the amorphous or crystalline form and excipient stabilizer in a appropriate solvent to form a liquid solution, and eliminating the solvent; and (3) a pharmaceutical composition comprising the amorphous solid solution.
IPC 8 full level
C07D 231/14 (2006.01); A61K 31/415 (2006.01)
CPC (source: EP KR US)
A61K 31/415 (2013.01 - KR); A61P 3/04 (2017.12 - EP); A61P 3/06 (2017.12 - EP); A61P 25/00 (2017.12 - EP); C07D 231/14 (2013.01 - EP KR US); C07D 401/04 (2013.01 - KR)
Citation (search report)
See references of WO 2008129157A2
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA MK RS
DOCDB simple family (publication)
FR 2913018 A1 20080829; AR 065410 A1 20090603; AU 2008240507 A1 20081030; BR PI0807575 A2 20140701; CA 2678801 A1 20081030; CL 2008000550 A1 20080704; CN 101641333 A 20100203; CO 6210812 A2 20101020; EA 200970792 A1 20100430; EP 2132182 A2 20091216; IL 200370 A0 20100429; JP 2010519246 A 20100603; KR 20090113305 A 20091029; MA 31244 B1 20100301; MX 2009008991 A 20090903; PE 20081778 A1 20090101; TW 200846339 A 20081201; US 2010076023 A1 20100325; UY 30937 A1 20080930; WO 2008129157 A2 20081030; WO 2008129157 A3 20081231; WO 2008129157 A4 20090305
DOCDB simple family (application)
FR 0701377 A 20070223; AR P080100705 A 20080221; AU 2008240507 A 20080220; BR PI0807575 A 20080220; CA 2678801 A 20080220; CL 2008000550 A 20080222; CN 200880009562 A 20080220; CO 09087002 A 20090819; EA 200970792 A 20080220; EP 08775573 A 20080220; FR 2008000216 W 20080220; IL 20037009 A 20090812; JP 2009550302 A 20080220; KR 20097017532 A 20080220; MA 32210 A 20090910; MX 2009008991 A 20080220; PE 2008000359 A 20080220; TW 97106126 A 20080221; US 54394209 A 20090819; UY 30937 A 20080222