EP 2146990 A1 20100127 - TRIAZOLOPYRIDINE CARBOXAMIDE DERIVATIVES AND TRIAZOLOPYRIMIDINE CARBOXAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
Title (en)
TRIAZOLOPYRIDINE CARBOXAMIDE DERIVATIVES AND TRIAZOLOPYRIMIDINE CARBOXAMIDE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
Title (de)
TRIAZOLPYRIDIN-CARBOXAMID-DERIVATE UND TRIAZOLPYRIMIDIN-CARBOXAMID-DERIVATE, IHRE HERSTELLUNG UND IHRE THERAPEUTISCHE ANWENDUNG
Title (fr)
DÉRIVÉS DE TRIAZOLOPYRIDINE-CARBOXAMIDES ET TRIAZOLOPYRIMIDINE-CARBOXAMIDES, LEUR PRÉPARATION ET LEUR APPLICATION EN THÉRAPEUTIQUE
Publication
Application
Priority
- FR 2008000532 W 20080416
- FR 0702809 A 20070418
Abstract (en)
[origin: WO2008145839A1] The invention relates to the triazolopyridine carboxamide derivatives and triazolopyrimidine carboxamide derivatives of general formula (I) in which: A and X are, independently of one another, a nitrogen atom or a CH group; R1 is an NR3R4 group, in which R3 and R4 form, with the nitrogen atom which bears them, a heterocyclic group comprising 3 to 7 ring members that may incorporate an oxygen or sulphur atom, an NR group or an NR'-CO group, wherein said ring is optionally substituted with one or more groups selected from a halogen atom or a (C1-C6)alkyl, (C1-C6)alkoxy, halo(C1-C6)alkyl or halo(C1- C6)alkoxy group, R2 is an aryl group, optionally substituted with one or more groups selected from a halogen atom or a methyl, trifluoromethyl, methoxy or trifluoromethoxy group. Process for the preparation thereof and therapeutic use thereof.
IPC 8 full level
C07D 471/04 (2006.01); A61K 31/4439 (2006.01); A61P 37/00 (2006.01); C07D 487/04 (2006.01)
CPC (source: EP KR US)
A61K 31/4439 (2013.01 - KR); A61P 1/00 (2017.12 - EP); A61P 1/04 (2017.12 - EP); A61P 1/08 (2017.12 - EP); A61P 1/12 (2017.12 - EP); A61P 3/00 (2017.12 - EP); A61P 3/04 (2017.12 - EP); A61P 3/06 (2017.12 - EP); A61P 7/06 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/06 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 9/12 (2017.12 - EP); A61P 11/00 (2017.12 - EP); A61P 11/06 (2017.12 - EP); A61P 13/00 (2017.12 - EP); A61P 13/10 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 17/00 (2017.12 - EP); A61P 17/06 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 19/06 (2017.12 - EP); A61P 19/10 (2017.12 - EP); A61P 21/00 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/02 (2017.12 - EP); A61P 25/04 (2017.12 - EP); A61P 25/06 (2017.12 - EP); A61P 25/08 (2017.12 - EP); A61P 25/14 (2017.12 - EP); A61P 25/16 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 25/20 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 27/00 (2017.12 - EP); A61P 27/02 (2017.12 - EP); A61P 27/06 (2017.12 - EP); A61P 27/16 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 31/00 (2017.12 - EP); A61P 31/04 (2017.12 - EP); A61P 31/12 (2017.12 - EP); A61P 31/18 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 37/00 (2017.12 - EP); A61P 37/02 (2017.12 - EP); A61P 37/06 (2017.12 - EP); A61P 37/08 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 471/04 (2013.01 - EP KR US); C07D 487/04 (2013.01 - EP KR US)
Citation (search report)
See references of WO 2008145839A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA MK RS
DOCDB simple family (publication)
FR 2915199 A1 20081024; FR 2915199 B1 20100122; AR 066107 A1 20090722; AU 2008257320 A1 20081204; BR PI0810440 A2 20141014; CA 2683929 A1 20081204; CL 2008001104 A1 20090116; CN 101668758 A 20100310; EP 2146990 A1 20100127; IL 201450 A0 20100531; JP 2010524904 A 20100722; KR 20090130057 A 20091217; MX 2009011212 A 20091102; RU 2009142431 A 20110527; TW 200901993 A 20090116; US 2010041651 A1 20100218; US 8080547 B2 20111220; UY 31032 A1 20081128; WO 2008145839 A1 20081204; WO 2008145839 A8 20091119
DOCDB simple family (application)
FR 0702809 A 20070418; AR P080101601 A 20080418; AU 2008257320 A 20080416; BR PI0810440 A 20080416; CA 2683929 A 20080416; CL 2008001104 A 20080417; CN 200880012545 A 20080416; EP 08787961 A 20080416; FR 2008000532 W 20080416; IL 20145009 A 20091011; JP 2010503547 A 20080416; KR 20097021591 A 20080416; MX 2009011212 A 20080416; RU 2009142431 A 20080416; TW 97114018 A 20080417; US 57395909 A 20091006; UY 31032 A 20080418