Global Patent Index - EP 2149549 A4

EP 2149549 A4 20120104 - PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF HEPATITIS

Title (en)

PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF HEPATITIS

Title (de)

PHARMAZEUTISCHE ZUSAMMENSETZUNG ZUR PRÄVENTION ODER BEHANDLUNG VON HÄPATITIS

Title (fr)

COMPOSITION PHARMACEUTIQUE DESTINÉE À LA PRÉVENTION OU AU TRAITEMENT DE L'HÉPATITE

Publication

EP 2149549 A4 20120104 (EN)

Application

EP 08764487 A 20080522

Priority

  • JP 2008059414 W 20080522
  • JP 2007138771 A 20070525

Abstract (en)

[origin: EP2149549A1] The present invention provides a pharmaceutical composition for prophylaxis or treatment of hepatitis. Solution A pharmaceutical composition for prophylaxis or treatment of hepatitis, comprising a compound represented by the general formula (I): wherein R 1 represents a C 1 -C 4 alkyl group, R 2 and R 3 which are the same or different represent a hydrogen atom, a C 1 -C 4 alkyl group, or a C 1 -C 4 alkoxy group, X represents a sulfur atom or a nitrogen atom substituted by a methyl group, and n represents an integer of 3 or 4, or a pharmacologically acceptable salt thereof as an active ingredient.

IPC 8 full level

C07D 207/335 (2006.01); A61K 31/381 (2006.01); A61K 31/40 (2006.01); A61P 1/16 (2006.01); A61P 37/06 (2006.01); C07D 333/22 (2006.01)

CPC (source: EP US)

A61K 31/381 (2013.01 - EP US); A61K 31/404 (2013.01 - EP US); A61P 1/04 (2017.12 - EP); A61P 1/16 (2017.12 - EP); A61P 17/06 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 31/12 (2017.12 - EP); A61P 37/06 (2017.12 - EP); C07D 207/335 (2013.01 - EP US); C07D 333/22 (2013.01 - EP US); Y02A 50/30 (2017.12 - EP US)

Citation (search report)

  • [X] WO 2006137509 A1 20061228 - SANKYO CO [JP], et al & EP 1915994 A1 20080430 - SANKYO CO [JP]
  • [X] EP 1733724 A1 20061220 - SANKYO CO [JP]
  • [X] EP 1300405 A1 20030409 - SANKYO CO [JP]
  • [X] DATABASE WPI Week 200512, Derwent World Patents Index; AN 2005-112609, XP002664222
  • [X] DATABASE WPI Week 200651, Derwent World Patents Index; AN 2006-497365, XP002664223
  • [A] MALEKZADEH R ET AL: "Cyclosporin A is a promising alternative to corticosteroids in autoimmune hepatitis.", June 2001, DIGESTIVE DISEASES AND SCIENCES JUN 2001 LNKD- PUBMED:11414311, VOL. 46, NR. 6, PAGE(S) 1321 - 1327, ISSN: 0163-2116, XP002664224
  • See references of WO 2008146691A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR

DOCDB simple family (publication)

EP 2149549 A1 20100203; EP 2149549 A4 20120104; JP WO2008146691 A1 20100819; TW 200906389 A 20090216; US 2010081702 A1 20100401; WO 2008146691 A1 20081204

DOCDB simple family (application)

EP 08764487 A 20080522; JP 2008059414 W 20080522; JP 2009516274 A 20080522; TW 97118598 A 20080521; US 62421409 A 20091123