Global Patent Index - EP 2150238 A1

EP 2150238 A1 20100210 - METHOD FOR THE PRODUCTION OF ADSORBATES OF A RASAGILINE SALT HAVING A WATER SOLUBLE ADJUVANT

Title (en)

METHOD FOR THE PRODUCTION OF ADSORBATES OF A RASAGILINE SALT HAVING A WATER SOLUBLE ADJUVANT

Title (de)

HERSTELLUNGSVERFAHREN FÜR ADSORBATE EINES RASAGILINSALZES MIT EINEM WASSERLÖSLICHEN HILFSSTOFF

Title (fr)

PROCÉDÉ DE PRÉPARATION D'ADSORBATS D'UN SEL DE RASAGILINE COMPRENANT UNE SUBSTANCE AUXILIAIRE SOLUBLE DANS L'EAU

Publication

EP 2150238 A1 20100210 (DE)

Application

EP 08749245 A 20080430

Priority

  • EP 2008003498 W 20080430
  • EP 07008755 A 20070430
  • EP 08749245 A 20080430

Abstract (en)

[origin: EP1987816A1] Adsorbate production involves spray drying of a solution of a pharmaceutical compatible salt of the rasagiline and a pharmaceutical compatible, water-soluble and organic adjuvant. The pharmaceutical compatible salt of the rasagilins is a mesylate salt. One or multiple pharmaceutical compatibles, water-soluble or water-insoluble e.g. micro-crystalline cellulose are also provided.

IPC 8 full level

A61K 9/16 (2006.01); A61K 9/20 (2006.01); A61K 31/00 (2006.01)

CPC (source: EP US)

A61K 9/1629 (2013.01 - EP US); A61K 9/1635 (2013.01 - EP US); A61K 9/1652 (2013.01 - EP US); A61K 9/1694 (2013.01 - EP US); A61K 9/2054 (2013.01 - EP US); A61K 9/2059 (2013.01 - EP US); A61K 9/2095 (2013.01 - EP US); A61K 31/135 (2013.01 - EP US); A61K 47/542 (2017.07 - EP US); A61K 47/58 (2017.07 - EP US); A61K 47/61 (2017.07 - EP US); A61P 25/16 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 25/28 (2017.12 - EP)

Citation (search report)

See references of WO 2008131961A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA MK RS

DOCDB simple family (publication)

EP 1987816 A1 20081105; CA 2684977 A1 20081106; CA 2684977 C 20150224; EP 2150238 A1 20100210; US 2010137447 A1 20100603; US 2014072526 A1 20140313; WO 2008131961 A1 20081106

DOCDB simple family (application)

EP 07008755 A 20070430; CA 2684977 A 20080430; EP 08749245 A 20080430; EP 2008003498 W 20080430; US 201314016960 A 20130903; US 59830108 A 20080430