Global Patent Index - EP 2170835 A1

EP 2170835 A1 20100407 - PROCESS FOR PREPARING TELMISARTAN

Title (en)

PROCESS FOR PREPARING TELMISARTAN

Title (de)

VERFAHREN ZUR HERSTELLUNG VON TELMISARTAN

Title (fr)

PROCÉDÉ DE PRÉPARATION DE TELMISARTAN

Publication

EP 2170835 A1 20100407 (EN)

Application

EP 08774728 A 20080703

Priority

  • EP 2008058616 W 20080703
  • SI 200700161 A 20070703
  • SI 200700322 A 20071210

Abstract (en)

[origin: WO2009004064A1] Novel processes for preparing a telmisaitan nitrile intermediate (4'-[{2-n-propyl-4- methyI-6-f l-methyJbenzimidazol-2-yl)-benzimidazol- l -yl)-methyl]-biphenyl-2-nitrile) and further converting it to telmisaitan and/or salts thereof are disclosed.

IPC 8 full level

C07D 235/08 (2006.01); A61K 31/4184 (2006.01); A61P 9/12 (2006.01); C07D 235/18 (2006.01); C07D 235/20 (2006.01)

CPC (source: EP)

A61P 9/12 (2017.12); C07D 235/08 (2013.01); C07D 235/18 (2013.01); C07D 235/20 (2013.01)

Citation (search report)

See references of WO 2009004064A1

Citation (examination)

WEI-ZHE XUE ET AL: "Synthesis of Telmisartan and Its Derivatives and Evaluation of Their Biological Activities", 2006 SIXTH CHINA PHARMACEUTICAL ASSOCIATION ANNUAL CONFERENCE PROCEEDINGS; NOVEMBER 2006; GUANGZHOU, CHINA, 1 January 2006 (2006-01-01) - November 2006 (2006-11-01), CN, pages 1113 - 1118, XP055171125

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA MK RS

DOCDB simple family (publication)

WO 2009004064 A1 20090108; CN 101743228 A 20100616; CN 101743228 B 20140129; EA 200901619 A1 20100430; EP 2170835 A1 20100407

DOCDB simple family (application)

EP 2008058616 W 20080703; CN 200880022887 A 20080703; EA 200901619 A 20080703; EP 08774728 A 20080703