EP 2173354 A1 20100414 - QUINOXALINE DERIVATIVES AS PI3 KINASE INHIBITORS
Title (en)
QUINOXALINE DERIVATIVES AS PI3 KINASE INHIBITORS
Title (de)
CHINOXALINDERIVATE ALS PI3-KINASE-INHIBITOREN
Title (fr)
DÉRIVÉS DES QUINOXALINES UTILISÉS COMME INHIBITEURS DES PI3-KINASES
Publication
Application
Priority
- US 2008072401 W 20080807
- US 95484507 P 20070809
Abstract (en)
[origin: WO2009021083A1] Invented is a method of inhibiting the activity/function of PI3 kinases using quinoxaline derivatives. Also invented is a method of treating one or more disease states selected from: autoimmune disorders, inflammatory diseases, cardiovascular diseases, neurodegenerative diseases, allergy, asthma, pancreatitis, multiorgan failure, kidney diseases, platelet aggregation, cancer, sperm motility, transplantation rejection, graft rejection and lung injuries by the administration of quinoxaline derivatives.
IPC 8 full level
A61K 31/535 (2006.01); A61P 35/00 (2006.01); C07D 401/14 (2006.01); C07D 403/04 (2006.01); C07D 403/14 (2006.01); C07D 405/04 (2006.01); C07D 405/14 (2006.01); C07D 413/14 (2006.01); C07D 471/04 (2006.01); C07D 495/04 (2006.01)
CPC (source: EP)
A61P 1/04 (2017.12); A61P 1/18 (2017.12); A61P 7/02 (2017.12); A61P 9/04 (2017.12); A61P 9/10 (2017.12); A61P 9/12 (2017.12); A61P 11/00 (2017.12); A61P 11/06 (2017.12); A61P 13/12 (2017.12); A61P 15/08 (2017.12); A61P 17/02 (2017.12); A61P 17/06 (2017.12); A61P 19/02 (2017.12); A61P 25/00 (2017.12); A61P 25/14 (2017.12); A61P 25/28 (2017.12); A61P 29/00 (2017.12); A61P 31/04 (2017.12); A61P 35/00 (2017.12); A61P 35/02 (2017.12); A61P 35/04 (2017.12); A61P 37/00 (2017.12); A61P 37/06 (2017.12); A61P 37/08 (2017.12); A61P 43/00 (2017.12); C07D 401/14 (2013.01); C07D 403/04 (2013.01); C07D 403/14 (2013.01); C07D 405/04 (2013.01); C07D 405/14 (2013.01); C07D 413/14 (2013.01); C07D 471/04 (2013.01); C07D 495/04 (2013.01)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA MK RS
DOCDB simple family (publication)
WO 2009021083 A1 20090212; WO 2009021083 A8 20090409; EP 2173354 A1 20100414; EP 2173354 A4 20111005; JP 2010535804 A 20101125
DOCDB simple family (application)
US 2008072401 W 20080807; EP 08797323 A 20080807; JP 2010520295 A 20080807