EP 2185560 A1 20100519 - HETEROARYL AMIDE ANALOGUES
Title (en)
HETEROARYL AMIDE ANALOGUES
Title (de)
HETEROARYLAMIDANALOGE
Title (fr)
ANALOGUES D'HÉTÉROARYLAMIDES
Publication
Application
Priority
- US 2008072760 W 20080811
- US 95525007 P 20070810
Abstract (en)
[origin: WO2009023623A1] Compounds, pharmaceutical compositions, and methods of use are disclosed for heteroaryl amide analogues of formula Ia and/or Ib: . In certain embodiments, the heteroaryl amide analogues are agonists and/or ligands of dopamine receptors and may be useful, inter alia, for the treatment of a condition responsive to P2X7 receptor modulation, for example, pain, inflammation, a neurological or neurodegenerative disorder, a cardiovascular disorder, an ocular disorder or an immune system disorder.
IPC 8 full level
C07D 401/04 (2006.01); A61K 31/506 (2006.01); A61P 25/02 (2006.01); C07D 401/12 (2006.01); C07D 401/14 (2006.01); C07D 403/04 (2006.01); C07D 471/04 (2006.01)
CPC (source: EP KR)
A61P 1/16 (2017.12 - EP); A61P 11/00 (2017.12 - EP); A61P 11/06 (2017.12 - EP); A61P 25/02 (2017.12 - EP); A61P 25/04 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 27/02 (2017.12 - EP); A61P 27/06 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 401/04 (2013.01 - EP); C07D 401/12 (2013.01 - EP); C07D 401/14 (2013.01 - EP); C07D 403/04 (2013.01 - EP KR); C07D 471/04 (2013.01 - EP); C07D 487/04 (2013.01 - KR)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA MK RS
DOCDB simple family (publication)
WO 2009023623 A1 20090219; AU 2008286946 A1 20090219; AU 2008286946 B2 20131121; BR PI0812594 A2 20150623; CA 2691512 A1 20090219; CN 101778850 A 20100714; CO 6251319 A2 20110221; EA 020332 B1 20141030; EA 200971085 A1 20100630; EP 2185560 A1 20100519; EP 2185560 A4 20111005; IL 202550 A0 20100630; JP 2010535816 A 20101125; JP 2015110566 A 20150618; KR 20100066422 A 20100617; NZ 582056 A 20120831; SG 183699 A1 20120927; UA 99729 C2 20120925
DOCDB simple family (application)
US 2008072760 W 20080811; AU 2008286946 A 20080811; BR PI0812594 A 20080811; CA 2691512 A 20080811; CN 200880021498 A 20080811; CO 09146587 A 20091222; EA 200971085 A 20080811; EP 08797591 A 20080811; IL 20255009 A 20091206; JP 2010520343 A 20080811; JP 2014238138 A 20141125; KR 20097026704 A 20080811; NZ 58205608 A 20080811; SG 2012058533 A 20080811; UA A200913336 A 20080811