EP 2200998 A1 20100630 - AZACYCLYLISOQUINOLINONE AND ISOINDOLINONE DERIVATIVES AS HISTAMINE-3 ANTAGONISTS
Title (en)
AZACYCLYLISOQUINOLINONE AND ISOINDOLINONE DERIVATIVES AS HISTAMINE-3 ANTAGONISTS
Title (de)
AZACYCLYLISOCHINOLINON- UND ISOINDOLINONDERIVATE ALS HISTAMIN-3-ANTAGONISTEN
Title (fr)
DÉRIVÉS D'AZACYCLYLISOQUINOLINONE ET D'ISOINDOLINONE CONVENANT COMME ANTAGONISTES DE L'HISTAMINE-3
Publication
Application
Priority
- US 2008075942 W 20080911
- US 99355407 P 20070912
Abstract (en)
[origin: WO2009036117A1] The present invention provides a compound of formula (I) and the use thereof for the treatment of a central nervous system disorder related to or affected by the histamine-3 receptor.
IPC 8 full level
C07D 401/04 (2006.01); A61K 31/4025 (2006.01); A61K 31/435 (2006.01); A61P 25/00 (2006.01); C07D 401/14 (2006.01); C07D 403/04 (2006.01); C07D 403/14 (2006.01)
CPC (source: EP US)
A61P 9/00 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/14 (2017.12 - EP); A61P 25/16 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 401/04 (2013.01 - EP US); C07D 401/14 (2013.01 - EP US); C07D 403/04 (2013.01 - EP US); C07D 403/14 (2013.01 - EP US)
Citation (search report)
See references of WO 2009036117A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA MK RS
DOCDB simple family (publication)
WO 2009036117 A1 20090319; AP 2010005199 A0 20100430; AU 2008298983 A1 20090319; BR PI0816806 A2 20150310; CA 2699383 A1 20090319; CL 2008002708 A1 20081010; CN 101842366 A 20100922; CO 6300951 A2 20110721; CR 11309 A 20100407; DO P2010000078 A 20100415; EA 201000319 A1 20101029; EC SP10010032 A 20100831; EP 2200998 A1 20100630; JP 2010539178 A 20101216; KR 20100054852 A 20100525; MA 31700 B1 20100901; MX 2010002899 A 20100409; NI 201000035 A 20100715; PA 8795601 A1 20090515; PE 20090679 A1 20090528; TN 2010000107 A1 20110926; TW 200918062 A 20090501; US 2009069370 A1 20090312
DOCDB simple family (application)
US 2008075942 W 20080911; AP 2010005199 A 20080911; AU 2008298983 A 20080911; BR PI0816806 A 20080911; CA 2699383 A 20080911; CL 2008002708 A 20080911; CN 200880113557 A 20080911; CO 10030401 A 20100315; CR 11309 A 20100311; DO 2010000078 A 20100311; EA 201000319 A 20080911; EC SP10010032 A 20100312; EP 08830104 A 20080911; JP 2010524972 A 20080911; KR 20107007636 A 20080911; MA 32689 A 20100312; MX 2010002899 A 20080911; NI 201000035 A 20100311; PA 8795601 A 20080912; PE 2008001588 A 20080911; TN 2010000107 A 20100311; TW 97134761 A 20080910; US 20878008 A 20080911