Global Patent Index - EP 2227464 A1

EP 2227464 A1 20100915 - DERIVATIVES OF 1-[(IMIDAZOLIDIN-2-YL)IMINO)]INDAZOLE

Title (en)

DERIVATIVES OF 1-[(IMIDAZOLIDIN-2-YL)IMINO)]INDAZOLE

Title (de)

DERIVATE VON 1-[(IMIDAZOLIDIN-2-YL)IMINO]INDAZOL

Title (fr)

DÉRIVÉS DU 1-[(IMIDAZOLIDIN-2-YL)IMINO)]INDAZOLE

Publication

EP 2227464 A1 20100915 (EN)

Application

EP 08857024 A 20081205

Priority

  • GB 2008004024 W 20081205
  • PL 38395507 A 20071205

Abstract (en)

[origin: WO2009071906A1] The invention provides a compound of formula (I) wherein R1 denotes hydrogen, methyl or phenyl; R2, R3, R4 and R5 denote hydrogen, halogen, preferably a chlorine atom, alkyl, preferably methyl, alkoxyl, preferably methoxyl; m denotes a number 0 or 1; and HX denotes sulfuric, phosphoric, acetic, malonic, fumaric, oxalic, lactic, tartaric, citric, gluconic, p-toluenesulfonic, methanesulfonic acid, hydrogen bromide or hydrogen iodide, preferably hydrogen chloride. The use of the compounds as a2-adrenergic receptor agonists is also provided.

IPC 8 full level

A61K 31/4178 (2006.01); A61P 9/00 (2006.01); C07D 403/12 (2006.01)

CPC (source: EP)

A61P 1/06 (2017.12); A61P 1/12 (2017.12); A61P 9/00 (2017.12); A61P 9/12 (2017.12); A61P 21/02 (2017.12); A61P 25/30 (2017.12); A61P 25/32 (2017.12); A61P 25/36 (2017.12); A61P 27/06 (2017.12); A61P 29/00 (2017.12); A61P 33/00 (2017.12); C07D 403/12 (2013.01)

Citation (search report)

See references of WO 2009071906A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA MK RS

DOCDB simple family (publication)

WO 2009071906 A1 20090611; EP 2227464 A1 20100915; PL 212581 B1 20121031; PL 383955 A1 20090608

DOCDB simple family (application)

GB 2008004024 W 20081205; EP 08857024 A 20081205; PL 38395507 A 20071205