EP 2238131 A1 20101013 - 5-O-SUBSTITUTED 3-N-PHENYL-1,3,4-OXADIAZOLONES FOR MEDICAL USE
Title (en)
5-O-SUBSTITUTED 3-N-PHENYL-1,3,4-OXADIAZOLONES FOR MEDICAL USE
Title (de)
5-O-SUBSTITUIERTE 3-N-PHENYL-1,3,4-OXADIAZOLONE ZUR MEDIZINISCHEN VERWENDUNG
Title (fr)
3-N-PHÉNYL-1,3,4-OXADIAZOLONES 5-O-SUBSTITUÉES POUR UNE UTILISATION MÉDICALE
Publication
Application
Priority
- PT 2008000054 W 20081223
- US 930207 P 20071227
Abstract (en)
[origin: WO2009084970A1] The present invention relates to compounds having a 5-O-substituted 3-N-phenyl-1,3,4-oxadiazolone structural unit which have unexpectedly high level of inhibition of FAAH (fatty acid amide hydrolase). (I)
IPC 8 full level
C07D 413/10 (2006.01); A61K 31/4245 (2006.01); A61P 9/00 (2006.01); A61P 11/00 (2006.01); A61P 25/00 (2006.01); C07D 271/113 (2006.01); C07D 413/12 (2006.01)
CPC (source: EP)
A61P 1/00 (2017.12); A61P 1/04 (2017.12); A61P 1/08 (2017.12); A61P 3/10 (2017.12); A61P 9/00 (2017.12); A61P 11/00 (2017.12); A61P 19/00 (2017.12); A61P 19/02 (2017.12); A61P 19/06 (2017.12); A61P 19/10 (2017.12); A61P 25/00 (2017.12); A61P 25/08 (2017.12); A61P 25/20 (2017.12); A61P 25/28 (2017.12); A61P 27/02 (2017.12); A61P 29/00 (2017.12); A61P 31/04 (2017.12); A61P 31/12 (2017.12); A61P 33/00 (2017.12); A61P 35/00 (2017.12); A61P 37/00 (2017.12); A61P 43/00 (2017.12); C07D 271/113 (2013.01); C07D 413/10 (2013.01); C07D 413/12 (2013.01)
Citation (search report)
See references of WO 2009084970A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MT NL NO PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA MK RS
DOCDB simple family (publication)
WO 2009084970 A1 20090709; AR 069970 A1 20100303; AU 2008344032 A1 20090709; AU 2008344032 A8 20100819; BR PI0821482 A2 20150714; CA 2710743 A1 20090709; CL 2008003895 A1 20100625; CN 101959881 A 20110126; EP 2238131 A1 20101013; IL 206419 A0 20101230; JP 2011507952 A 20110310; KR 20100111691 A 20101015; MX 2010006995 A 20100818; TW 200932732 A 20090801; ZA 201005306 B 20110428
DOCDB simple family (application)
PT 2008000054 W 20081223; AR P080105707 A 20081223; AU 2008344032 A 20081223; BR PI0821482 A 20081223; CA 2710743 A 20081223; CL 2008003895 A 20081223; CN 200880127681 A 20081223; EP 08866782 A 20081223; IL 20641910 A 20100616; JP 2010540610 A 20081223; KR 20107015516 A 20081223; MX 2010006995 A 20081223; TW 97150238 A 20081223; ZA 201005306 A 20100726