EP 2252372 A1 20101124 - 2-AMINOQUINOLINES
Title (en)
2-AMINOQUINOLINES
Title (de)
2-AMINOCHINOLINE
Title (fr)
2-AMINOQUINOLÉINES
Publication
Application
Priority
- EP 2009052253 W 20090226
- EP 08152425 A 20080307
- EP 09718263 A 20090226
Abstract (en)
[origin: US2009227583A1] The present invention relates to compounds of formula (I) wherein A, R1, R2, R3, R4, and R5 are as described herein, pharmaceutical compositions containing them, and methods for their manufacture. These compounds are 5-HT5A receptor antagonistsand are useful in the prevention and/or treatment of depression, anxiety disorders, schizophrenia, panic disorders, agoraphobia, social phobia, obsessive compulsive disorders, post-traumatic stress disorders, pain, memory disorders, dementia, disorders of eating behaviors, sexual dysfunction, sleep disorders, abuse of drugs, motor disorders such as Parkinson's disease, psychiatric disorders or gastrointestinal disorders.
IPC 8 full level
A61P 25/00 (2006.01); A61K 31/47 (2006.01); A61K 31/4709 (2006.01); C07D 215/38 (2006.01); C07D 401/04 (2006.01); C07D 405/12 (2006.01); C07D 405/14 (2006.01); C07D 413/04 (2006.01)
CPC (source: EP US)
A61P 1/04 (2017.12 - EP); A61P 15/10 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/04 (2017.12 - EP); A61P 25/14 (2017.12 - EP); A61P 25/16 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 25/20 (2017.12 - EP); A61P 25/22 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 25/30 (2017.12 - EP); A61P 25/32 (2017.12 - EP); A61P 25/34 (2017.12 - EP); A61P 25/36 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 215/38 (2013.01 - EP US); C07D 401/04 (2013.01 - EP US); C07D 401/12 (2013.01 - EP US); C07D 405/14 (2013.01 - EP US); C07D 409/12 (2013.01 - EP US); C07D 413/12 (2013.01 - EP US); C07D 413/14 (2013.01 - EP US); C07D 417/12 (2013.01 - EP US)
Citation (search report)
See references of WO 2009109502A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA RS
DOCDB simple family (publication)
US 2009227583 A1 20090910; US 8188284 B2 20120529; AU 2009221294 A1 20090911; BR PI0909824 A2 20190306; CA 2711247 A1 20090911; CN 101939055 A 20110105; EP 2252372 A1 20101124; IL 206761 A0 20101230; JP 2011513353 A 20110428; KR 20100119789 A 20101110; MX 2010008239 A 20100818; WO 2009109502 A1 20090911
DOCDB simple family (application)
US 39407209 A 20090227; AU 2009221294 A 20090226; BR PI0909824 A 20090226; CA 2711247 A 20090226; CN 200980104695 A 20090226; EP 09718263 A 20090226; EP 2009052253 W 20090226; IL 20676110 A 20100701; JP 2010549101 A 20090226; KR 20107019839 A 20090226; MX 2010008239 A 20090226