EP 2260037 A2 20101215 - A POLYMORPHIC FORM OF A PYRAZINO [2,3-H] [3] BENZAZEPINE DERIVATIVE
Title (en)
A POLYMORPHIC FORM OF A PYRAZINO [2,3-H] [3] BENZAZEPINE DERIVATIVE
Title (de)
POLYMORPHE FORM EINES PYRAZINO[2,3-H][3]BENZAZEPINDERIVATS
Title (fr)
NOUVELLE FORME POLYMORPHE D'UN DÉRIVÉ DE PYRAZINO[2,3-H][3]-BENZAZÉPINE
Publication
Application
Priority
- EP 2009051727 W 20090213
- US 6603208 P 20080215
Abstract (en)
[origin: WO2009101185A2] The invention relates generally to a crystalline polymorphic form of 7, 8, 9, 10-tetrahydro-6, 10-methano-6H-pyrazino[2, 3-h][3] benzazepine, varenicline base, i.e. a hydrate of varenicline base, designated herein as Form II, and to a method for preparing and obtaining the same.
IPC 8 full level
A61P 25/34 (2006.01); C07D 471/08 (2006.01)
CPC (source: EP)
A61P 25/34 (2017.12); C07D 471/08 (2013.01)
Citation (search report)
See references of WO 2009101185A2
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR
Designated extension state (EPC)
AL BA RS
DOCDB simple family (publication)
WO 2009101185 A2 20090820; WO 2009101185 A3 20091203; EP 2260037 A2 20101215
DOCDB simple family (application)
EP 2009051727 W 20090213; EP 09709821 A 20090213