Global Patent Index - EP 2271644 A1

EP 2271644 A1 20110112 - SUBSTITUTED PIPERIDINES AS THERAPEUTIC COMPOUNDS

Title (en)

SUBSTITUTED PIPERIDINES AS THERAPEUTIC COMPOUNDS

Title (de)

SUBSTITUIERTE PIPERIDINE ALS THERAPEUTISCHE ZUSAMMENSETZUNGEN

Title (fr)

PIPÉRIDINES SUBSTITUÉES À TITRE DE COMPOSÉS THÉRAPEUTIQUES

Publication

EP 2271644 A1 20110112 (EN)

Application

EP 09728288 A 20090401

Priority

  • EP 2009053898 W 20090401
  • EP 08153929 A 20080402
  • EP 09728288 A 20090401

Abstract (en)

[origin: WO2009121914A1] Described are compounds of the general formula (I), and pharmaceutically acceptable salt thereof, in which R1 has the definitions illustrated in detail in the description, as beta-secretase, cathepsin D, plasmepsin II and/or HIV protease inhibitors.

IPC 8 full level

C07D 413/12 (2006.01); A61K 31/5377 (2006.01); A61P 25/28 (2006.01); A61P 31/18 (2006.01); A61P 33/06 (2006.01)

CPC (source: EP)

A61P 25/28 (2017.12); A61P 31/18 (2017.12); A61P 33/06 (2017.12); A61P 43/00 (2017.12); C07D 413/12 (2013.01)

Citation (search report)

See references of WO 2009121914A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA RS

DOCDB simple family (publication)

WO 2009121914 A1 20091008; AU 2009232012 A1 20091008; BR PI0910991 A2 20160119; CA 2719070 A1 20091008; CN 101970431 A 20110209; EA 201001517 A1 20110429; EP 2271644 A1 20110112; JP 2011516453 A 20110526; KR 20110002459 A 20110107; MX 2010010876 A 20101026

DOCDB simple family (application)

EP 2009053898 W 20090401; AU 2009232012 A 20090401; BR PI0910991 A 20090401; CA 2719070 A 20090401; CN 200980108313 A 20090401; EA 201001517 A 20090401; EP 09728288 A 20090401; JP 2011502382 A 20090401; KR 20107022007 A 20090401; MX 2010010876 A 20090401