EP 2289868 B1 20140813 - CARBOXYLIC ACID COMPOUND
Title (en)
CARBOXYLIC ACID COMPOUND
Title (de)
CARBOXYLSÄUREVERBINDUNG
Title (fr)
COMPOSÉ D ACIDE CARBOXYLIQUE
Publication
Application
Priority
- JP 2009061350 W 20090623
- JP 2008165756 A 20080625
Abstract (en)
[origin: EP2289868A1] To find a therapeutic agent and/or a preventive agent for diabetes mellitus or the like having excellent activity and safety. A compound represented by the following general formula (I), or a pharmacologically acceptable salt thereof. In the formula, X represents =C(R5)- or =N-; Y represents -O- or -NH-; L represents a bond or a substitutable C1-C3 alkylene group; M represents a substitutable C3-C10 cycloalkyl group, a substitutable C6-C10 aryl group, or a substitutable heterocyclic group; R 1 represents a C1-C6 alkyl group, a C3-C10 cycloalkyl group, a C1-C6 haloalkyl group, a C1-C6 alkenyl group, a C1-C6 alkynyl group, a C1-C6 aliphatic acyl group, a C1-C6 alkoxy C1-C6 alkyl group, or a C6-C10 aryl group; and R 2 , R 3 , R 4 , and R 5 may be the same or different and each represent a hydrogen atom, a halogen atom, a C1-C3 alkyl group, a C1-C3 haloalkyl group, a C1-C3 alkoxy group, or a nitro group. In this connection, the alkyl group moieties of R 1 and R 2 may be bonded to each other to form a 5- to 6-membered heterocyclic ring containing one oxygen atom.
IPC 8 full level
C07C 59/66 (2006.01); A61K 31/192 (2006.01); A61K 31/195 (2006.01); A61P 1/14 (2006.01); C07C 59/72 (2006.01); C07C 205/34 (2006.01); C07C 205/37 (2006.01); C07C 217/76 (2006.01); C07C 229/42 (2006.01); C07C 255/54 (2006.01); C07C 311/29 (2006.01); C07C 317/22 (2006.01); C07D 207/325 (2006.01); C07D 215/22 (2006.01); C07D 249/04 (2006.01); C07D 277/24 (2006.01); C07D 277/64 (2006.01); C07D 307/83 (2006.01); C07D 491/048 (2006.01)
CPC (source: EP US)
A61K 31/192 (2013.01 - EP US); A61K 31/195 (2013.01 - EP US); A61K 31/196 (2013.01 - EP US); A61K 31/275 (2013.01 - EP US); A61K 31/343 (2013.01 - EP US); A61K 31/40 (2013.01 - EP US); A61K 31/4192 (2013.01 - EP US); A61K 31/426 (2013.01 - EP US); A61K 31/428 (2013.01 - EP US); A61K 31/47 (2013.01 - EP US); A61K 31/4741 (2013.01 - EP US); A61P 1/14 (2017.12 - EP); A61P 3/04 (2017.12 - EP); A61P 3/06 (2017.12 - EP); A61P 3/08 (2017.12 - EP); A61P 3/10 (2017.12 - EP); A61P 5/50 (2017.12 - EP); A61P 7/02 (2017.12 - EP); A61P 7/10 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 9/12 (2017.12 - EP); A61P 15/00 (2017.12 - EP); A61P 17/00 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 19/08 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 37/08 (2017.12 - EP); C07C 59/66 (2013.01 - EP US); C07C 59/72 (2013.01 - EP US); C07C 205/34 (2013.01 - EP US); C07C 205/37 (2013.01 - EP US); C07C 217/76 (2013.01 - EP US); C07C 229/42 (2013.01 - EP US); C07C 255/54 (2013.01 - EP US); C07C 311/29 (2013.01 - EP US); C07C 317/22 (2013.01 - EP US); C07D 207/325 (2013.01 - EP US); C07D 215/22 (2013.01 - EP US); C07D 249/04 (2013.01 - EP US); C07D 277/24 (2013.01 - EP US); C07D 277/64 (2013.01 - EP US); C07D 307/83 (2013.01 - EP US); C07D 491/048 (2013.01 - EP US); C07C 2601/02 (2017.04 - EP US); C07C 2602/08 (2017.04 - EP US)
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR
DOCDB simple family (publication)
EP 2289868 A1 20110302; EP 2289868 A4 20111207; EP 2289868 B1 20140813; AU 2009263384 A1 20091230; BR PI0913368 A2 20151124; CA 2727340 A1 20091230; CN 102076650 A 20110525; CO 6280528 A2 20110520; ES 2516716 T3 20141031; HK 1153453 A1 20120330; IL 210246 A0 20110331; JP 5425772 B2 20140226; JP WO2009157418 A1 20111215; KR 20110027657 A 20110316; MX 2010014571 A 20110325; NZ 588983 A 20111125; RU 2011102560 A 20120727; TW 201004917 A 20100201; US 2011053974 A1 20110303; US 8222281 B2 20120717; WO 2009157418 A1 20091230; ZA 201008096 B 20110831
DOCDB simple family (application)
EP 09770128 A 20090623; AU 2009263384 A 20090623; BR PI0913368 A 20090623; CA 2727340 A 20090623; CN 200980125186 A 20090623; CO 10162533 A 20101227; ES 09770128 T 20090623; HK 11107658 A 20110722; IL 21024610 A 20101223; JP 2009061350 W 20090623; JP 2010518013 A 20090623; KR 20107025765 A 20090623; MX 2010014571 A 20090623; NZ 58898309 A 20090623; RU 2011102560 A 20090623; TW 98121093 A 20090624; US 89359210 A 20100929; ZA 201008096 A 20101111