Global Patent Index - EP 2307012 A1

EP 2307012 A1 20110413 - NITROGEN HETEROCYCLE DERIVATIVES AS PROTEASOME MODULATORS

Title (en)

NITROGEN HETEROCYCLE DERIVATIVES AS PROTEASOME MODULATORS

Title (de)

STICKSTOFF-HETEROZYKLUS-DERIVATE ALS PROTEASOM-MODULATOREN

Title (fr)

DÉRIVÉS HÉTÉROCYCLIQUES DE L'AZOTE SOUS LA FORME DE MODULATEURS DU PROTÉASOME

Publication

EP 2307012 A1 20110413 (EN)

Application

EP 09773025 A 20090703

Priority

  • IB 2009052918 W 20090703
  • EP 08305377 A 20080704
  • EP 09773025 A 20090703

Abstract (en)

[origin: WO2010001365A1] The instant invention relates to the use of at least one nitrogen heterocycle derivative of formula (I): as proteasome activity modulator in the manufacture of a pharmaceutical composition intended to prevent and/or treat a disease condition mediated by the proteasome activity.

IPC 8 full level

A61K 31/4196 (2006.01); A61K 31/4245 (2006.01); A61P 9/10 (2006.01); A61P 29/00 (2006.01); A61P 31/04 (2006.01); A61P 31/12 (2006.01); A61P 33/06 (2006.01); A61P 35/00 (2006.01)

CPC (source: EP)

A61K 31/4196 (2013.01); A61K 31/4245 (2013.01); A61P 1/16 (2017.12); A61P 9/00 (2017.12); A61P 9/10 (2017.12); A61P 17/02 (2017.12); A61P 17/16 (2017.12); A61P 19/02 (2017.12); A61P 21/00 (2017.12); A61P 29/00 (2017.12); A61P 31/04 (2017.12); A61P 31/12 (2017.12); A61P 31/18 (2017.12); A61P 33/00 (2017.12); A61P 33/06 (2017.12); A61P 35/00 (2017.12); A61P 37/00 (2017.12); A61P 37/06 (2017.12); A61P 43/00 (2017.12); Y02A 50/30 (2017.12)

Citation (search report)

See references of WO 2010001365A1

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR

Designated extension state (EPC)

AL BA RS

DOCDB simple family (publication)

WO 2010001365 A1 20100107; CA 2728769 A1 20100107; EP 2307012 A1 20110413; JP 2011526620 A 20111013

DOCDB simple family (application)

IB 2009052918 W 20090703; CA 2728769 A 20090703; EP 09773025 A 20090703; JP 2011515719 A 20090703