Global Patent Index - EP 2331526 A2

EP 2331526 A2 20110615 - PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS

Title (en)

PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS

Title (de)

PYRIMIDINDERIVATE ALS KINASEINHIBITOREN

Title (fr)

DÉRIVÉS DE LA PYRIMIDINE COMME INHIBITEURS DE KINASES

Publication

EP 2331526 A2 20110615 (EN)

Application

EP 09770964 A 20090624

Priority

  • US 2009048509 W 20090624
  • US 7558308 P 20080625

Abstract (en)

[origin: WO2009158431A2] The invention provides novel pyrimidine derivatives and pharmaceutical compositions thereof, and methods for using such compounds. For example, the pyrimidine derivatives of the invention may be used to treat, ameliorate or prevent a condition which responds to inhibition of insulin-like growth factor (IGF-1R) or analplastic lymphoma kinase (ALK).

IPC 8 full level

C07D 401/14 (2006.01); A61K 31/506 (2006.01); A61P 31/00 (2006.01); A61P 35/00 (2006.01); A61P 37/00 (2006.01); C07D 403/12 (2006.01); C07D 403/14 (2006.01); C07D 405/14 (2006.01); C07D 409/14 (2006.01); C07D 413/14 (2006.01); C07D 417/14 (2006.01)

CPC (source: EP KR)

A61K 31/506 (2013.01 - KR); A61P 31/00 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 37/00 (2017.12 - EP); A61P 37/06 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 401/14 (2013.01 - EP); C07D 403/12 (2013.01 - EP KR); C07D 403/14 (2013.01 - EP); C07D 405/14 (2013.01 - EP); C07D 409/14 (2013.01 - EP); C07D 413/14 (2013.01 - EP KR); C07D 417/14 (2013.01 - EP)

Citation (search report)

See references of WO 2009158431A2

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK TR

Designated extension state (EPC)

AL BA RS

DOCDB simple family (publication)

WO 2009158431 A2 20091230; WO 2009158431 A3 20100311; AU 2009262198 A1 20091230; AU 2009262198 B2 20120927; BR PI0914545 A2 20170523; CA 2729546 A1 20091230; CN 102203083 A 20110928; EA 201100078 A1 20110830; EP 2331526 A2 20110615; JP 2011526291 A 20111006; KR 20110020940 A 20110303; MX 2010014568 A 20110329; UA 101057 C2 20130225

DOCDB simple family (application)

US 2009048509 W 20090624; AU 2009262198 A 20090624; BR PI0914545 A 20090624; CA 2729546 A 20090624; CN 200980129584 A 20090624; EA 201100078 A 20090624; EP 09770964 A 20090624; JP 2011516619 A 20090624; KR 20117001749 A 20090624; MX 2010014568 A 20090624; UA A201104068 A 20090624