Global Patent Index - EP 2346850 B1

EP 2346850 B1 20120905 - METHOD FOR THE PREPARATION OF DABIGATRAN AND ITS INTERMEDIATES

Title (en)

METHOD FOR THE PREPARATION OF DABIGATRAN AND ITS INTERMEDIATES

Title (de)

VERFAHREN ZUR HERSTELLUNG VON DABIGATRAN UND DESSEN ZWISCHENPRODUKTEN

Title (fr)

PROCÉDÉ POUR PRÉPARER LE DABIGATRAN ET SES INTERMÉDIAIRES

Publication

EP 2346850 B1 20120905 (EN)

Application

EP 09752269 A 20091026

Priority

  • CZ 2009000127 W 20091026
  • CZ 2008669 A 20081024

Abstract (en)

[origin: WO2010045900A1] Intermediates for the preparation of dabigatran of formulae (VII-2HC1) and (VII-HC1), methods for their preparation and a method for preparation of dabigatran of formula (VIII) using these intermediates.

IPC 8 full level

C07D 401/12 (2006.01)

CPC (source: EP US)

C07D 401/12 (2013.01 - EP US)

Designated contracting state (EPC)

AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR

DOCDB simple family (publication)

WO 2010045900 A1 20100429; CZ 2008669 A3 20100505; EA 018227 B1 20130628; EA 201100517 A1 20111031; EP 2346850 A1 20110727; EP 2346850 B1 20120905; ES 2393692 T3 20121227; SI 2346850 T1 20130131; UA 104438 C2 20140210; US 2011224441 A1 20110915; US 8394962 B2 20130312

DOCDB simple family (application)

CZ 2009000127 W 20091026; CZ 2008669 A 20081024; EA 201100517 A 20091026; EP 09752269 A 20091026; ES 09752269 T 20091026; SI 200930400 T 20091026; UA A201106447 A 20091026; US 200913124034 A 20091026