EP 2358369 A1 20110824 - Process for the preparation of substantially optically pure repaglinide and precursors thereof
Title (en)
Process for the preparation of substantially optically pure repaglinide and precursors thereof
Title (de)
VERFAHREN ZUR HERSTELLUNG VON WEITGEHEND OPTISCH REINEM REPAGLINID UND VORSTUFEN DAVON
Title (fr)
Procédé de synthèse de répaglinide substantiellement optiquement pure et de ses précurseurs
Publication
Application
Priority
- EP 2009063734 W 20091020
- EP 08167069 A 20081020
- EP 08173072 A 20081230
- EP 09154353 A 20090304
- EP 09737422 A 20091020
Abstract (en)
[origin: WO2010046360A1] The invention relates to a process for preparing substantially optically pure repaglinide and pharmaceutically acceptable salts, solvates and esters thereof. The invention further relates to a process for preparing precursors of repaglinide and in particular for preparing ( S ) ( f ) - 1 - ( 2 -piperidino-phenyl ) -3 - methyl - I -butylamine.
IPC 8 full level
A61K 31/4453 (2006.01); A61P 5/50 (2006.01); C07D 295/135 (2006.01)
CPC (source: EP)
A61P 5/50 (2017.12); C07D 295/135 (2013.01)
Citation (search report)
See references of WO 2010046360A1
Designated contracting state (EPC)
AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR
Designated extension state (EPC)
AL BA RS
DOCDB simple family (publication)
DOCDB simple family (application)
EP 2009063734 W 20091020; EP 09737422 A 20091020