EP 2526098 B1 20180711 - NITROGEN-CONTAINING HETEROARYL DERIVATIVES
Title (en)
NITROGEN-CONTAINING HETEROARYL DERIVATIVES
Title (de)
STICKSTOFFHALTIGE HETEROARYLDERIVATE
Title (fr)
DÉRIVÉS HÉTÉROARYLIQUES CONTENANT DE L'AZOTE
Publication
Application
Priority
- EP 10151364 A 20100122
- EP 2011050640 W 20110119
- EP 11701639 A 20110119
Abstract (en)
[origin: WO2011089132A1] The invention is concerned with novel nitrogen-containing heteroaryl derivatives of formula (I) wherein R1, R2, R3, R4, R5, A1, A2, and Y are as defined in the description and in the claims, as well as physiologically acceptable salts and esters thereof. These compounds inhibit PDE10A and can be used as medicaments.
IPC 8 full level
A61K 31/506 (2006.01); A61P 25/16 (2006.01); A61P 25/18 (2006.01); A61P 25/22 (2006.01); A61P 25/28 (2006.01); C07D 401/14 (2006.01); C07D 409/14 (2006.01); C07D 413/14 (2006.01); C07D 417/14 (2006.01)
CPC (source: EP KR US)
A61K 31/506 (2013.01 - KR); A61P 3/10 (2017.12 - EP); A61P 7/00 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 15/00 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 25/14 (2017.12 - EP); A61P 25/16 (2017.12 - EP); A61P 25/18 (2017.12 - EP); A61P 25/22 (2017.12 - EP); A61P 25/24 (2017.12 - EP); A61P 25/28 (2017.12 - EP); A61P 25/30 (2017.12 - EP); A61P 35/00 (2017.12 - EP); A61P 35/02 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 401/14 (2013.01 - EP KR US); C07D 409/14 (2013.01 - EP KR US); C07D 413/14 (2013.01 - EP US); C07D 417/14 (2013.01 - EP US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
WO 2011089132 A1 20110728; BR 112012017580 A2 20160816; CA 2782588 A1 20110728; CN 102712625 A 20121003; CN 102712625 B 20140409; EP 2526098 A1 20121128; EP 2526098 B1 20180711; HK 1171744 A1 20130405; JP 2013517316 A 20130516; JP 5735987 B2 20150617; KR 101734606 B1 20170511; KR 20120124454 A 20121113; MX 2012007536 A 20120730; RU 2012134306 A 20140227; RU 2559895 C2 20150820; US 2011183979 A1 20110728; US 8470820 B2 20130625
DOCDB simple family (application)
EP 2011050640 W 20110119; BR 112012017580 A 20110119; CA 2782588 A 20110119; CN 201180006401 A 20110119; EP 11701639 A 20110119; HK 12112511 A 20121205; JP 2012549340 A 20110119; KR 20127021841 A 20110119; MX 2012007536 A 20110119; RU 2012134306 A 20110119; US 201113005572 A 20110113