EP 2571362 A4 20140122 - IMPROVED PROCESS FOR A FOLATE-TARGETED AGENT
Title (en)
IMPROVED PROCESS FOR A FOLATE-TARGETED AGENT
Title (de)
VERBESSERTES VERFAHREN FÜR EIN FOLATANZIELUNGSMITTEL
Title (fr)
PROCÉDÉ PERFECTIONNÉ POUR UN AGENT FOLATE-CIBLÉ
Publication
Application
Priority
- US 201061351022 P 20100603
- US 34644410 P 20100519
- US 2011037134 W 20110519
IPC 8 full level
C07K 7/02 (2006.01); A61K 47/48 (2006.01)
CPC (source: EP)
A61K 47/551 (2017.07); C07K 7/02 (2013.01)
Citation (search report)
- [X] WO 2009002993 A1 20081231 - ENDOCYTE INC [US], et al
- [XD] WO 2007022493 A2 20070222 - ENDOCYTE INC [US], et al
- [X] VLAHOV I R ET AL: "Design and regioselective synthesis of a new generation of targeted chemotherapeutics. Part 1: EC145, a folic acid conjugate of desacetylvinblastine monohydrazide", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, GB, vol. 16, no. 19, 1 October 2006 (2006-10-01), pages 5093 - 5096, XP027966592, ISSN: 0960-894X, [retrieved on 20061001]
- See references of WO 2011146707A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
DOCDB simple family (application)
EP 11784235 A 20110519