Global Patent Index - EP 2632462 A1

EP 2632462 A1 2013-09-04 - NOVEL HETEROARYL-CARBOXAMIDE DERIVATIVES AS PDK1 INHIBITORS

Title (en)

NOVEL HETEROARYL-CARBOXAMIDE DERIVATIVES AS PDK1 INHIBITORS

Title (de)

NEUE HETEROARYL-CARBOXIMID-DERIVATE ALS PDK1-HEMMER

Title (fr)

NOUVEAUX DÉRIVÉS DE HÉTÉROARYL-CARBOXAMIDE UTILISÉS COMME INHIBITEURS DE LA PDK1

Publication

EP 2632462 A1 (EN)

Application

EP 11836931 A

Priority

  • US 40815910 P
  • US 2011057561 W

Abstract (en)

[origin: WO2012058176A1] This invention relates to certain Heteroaryl Carboxamide derivatives of Formula (I) as inhibitors of 3-phosphoinositide-dependent protein kinase (PDK-1). The compounds can be useful in inhibiting the proliferation of cancer cells, and other aberrant conditions where the PDK-1 signaling pathway is overstimulated.

IPC 8 full level (invention and additional information)

A61K 31/44 (2006.01); A61K 31/425 (2006.01); A61K 31/445 (2006.01)

CPC (invention and additional information)

A61K 31/425 (2013.01); A61K 31/445 (2013.01)

Citation (search report)

See references of WO 2012058176A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

EPO simple patent family

WO 2012058176 A1 20120503; EP 2632462 A1 20130904

INPADOC legal status


2013-11-20 [18W] APPLICATION WITHDRAWN

- Effective date: 20131017

2013-09-04 [17P] REQUEST FOR EXAMINATION FILED

- Effective date: 20130529

2013-09-04 [AK] DESIGNATED CONTRACTING STATES:

- Kind Code of Ref Document: A1

- Designated State(s): AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR