EP 2665719 B1 20160504 - FUSED DIHYDROFURANS AS GPR119 MODULATORS FOR THE TREATMENT OF DIABETES, OBESITY AND RELATED DISORDERS
Title (en)
FUSED DIHYDROFURANS AS GPR119 MODULATORS FOR THE TREATMENT OF DIABETES, OBESITY AND RELATED DISORDERS
Title (de)
KONDENSIERTE DIHYDROFURANE ALS GPR119-MODULATOREN ZUR BEHANDLUNG VON DIABETES, FETTLEIBIGKEIT UND VERWANDTEN ERKRANKUNGEN
Title (fr)
DIHYDROFURANES CONDENSÉS EN TANT QUE MODULATEURS DE GPR119 POUR LE TRAITEMENT DU DIABÈTE, DE L'OBÉSITÉ ET DE TROUBLES ASSOCIÉS
Publication
Application
Priority
- EP 11151688 A 20110121
- EP 11191903 A 20111205
- EP 2012050841 W 20120120
- EP 12700413 A 20120120
Abstract (en)
[origin: WO2012098217A1] The present invention relates to compounds of general formula (I), wherein the groups R1, LP, LQ, X1, X2, X3, A, n and m are as defined in the application, which have valuable pharmacological properties, and in particular bind to the GPR119 receptor and modulate its activity.
IPC 8 full level
A61K 31/454 (2006.01); A61K 31/4545 (2006.01); A61K 31/497 (2006.01); A61K 31/506 (2006.01); A61P 3/10 (2006.01); A61P 5/50 (2006.01); C07D 407/14 (2006.01); C07D 413/14 (2006.01); C07D 491/048 (2006.01)
CPC (source: EP KR US)
A61K 31/506 (2013.01 - KR); A61P 3/00 (2017.12 - EP); A61P 3/04 (2017.12 - EP); A61P 3/06 (2017.12 - EP); A61P 3/08 (2017.12 - EP); A61P 3/10 (2017.12 - EP); A61P 3/12 (2017.12 - EP); A61P 5/50 (2017.12 - EP); A61P 7/10 (2017.12 - EP); A61P 9/00 (2017.12 - EP); A61P 9/04 (2017.12 - EP); A61P 9/10 (2017.12 - EP); A61P 9/12 (2017.12 - EP); A61P 13/12 (2017.12 - EP); A61P 17/02 (2017.12 - EP); A61P 19/02 (2017.12 - EP); A61P 19/06 (2017.12 - EP); A61P 19/10 (2017.12 - EP); A61P 25/00 (2017.12 - EP); A61P 27/02 (2017.12 - EP); A61P 29/00 (2017.12 - EP); A61P 43/00 (2017.12 - EP); C07D 405/14 (2013.01 - KR); C07D 407/14 (2013.01 - EP US); C07D 413/14 (2013.01 - EP US); C07D 491/048 (2013.01 - EP US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2012098217 A1 20120726; AP 2013006985 A0 20130731; AR 084905 A1 20130710; AU 2012208530 A1 20130711; BR 112013017669 A2 20180918; CA 2825124 A1 20120726; CN 103443097 A 20131211; CO 6781501 A2 20131031; EA 201300846 A1 20131230; EC SP13012800 A 20131031; EP 2665719 A1 20131127; EP 2665719 B1 20160504; JP 2014502988 A 20140206; JP 5703393 B2 20150415; KR 20140003496 A 20140109; MA 34839 B1 20140102; MX 2013008083 A 20130913; SG 192036 A1 20130830; US 2013018030 A1 20130117; US 8778926 B2 20140715; UY 33871 A 20120731
DOCDB simple family (application)
EP 2012050841 W 20120120; AP 2013006985 A 20120120; AR P120100198 A 20120120; AU 2012208530 A 20120120; BR 112013017669 A 20120120; CA 2825124 A 20120120; CN 201280014027 A 20120120; CO 13177678 A 20130726; EA 201300846 A 20120120; EC SP13012800 A 20130729; EP 12700413 A 20120120; JP 2013549825 A 20120120; KR 20137019225 A 20120120; MA 36131 A 20130718; MX 2013008083 A 20120120; SG 2013055066 A 20120120; US 201213354356 A 20120120; UY 33871 A 20120120