Global Patent Index - EP 2665829 A1

EP 2665829 A1 20131127 - COMPOUNDS AND METHODS FOR THE IDENTIFICATION AND CHARACTERIZATION OF HDAC INTERACTING COMPOUNDS

Title (en)

COMPOUNDS AND METHODS FOR THE IDENTIFICATION AND CHARACTERIZATION OF HDAC INTERACTING COMPOUNDS

Title (de)

VERBINDUNGEN UND VERFAHREN ZUR IDENTIFIKATION UND CHARAKTERISIERUNG VON HDAC-INTERAGIERENDEN VERBINDUNGEN

Title (fr)

COMPOSÉS ET PROCÉDÉS POUR L'IDENTIFICATION ET LA CARACTÉRISATION DE COMPOSÉS INTERAGISSANT AVEC L'HDAC

Publication

EP 2665829 A1 20131127 (EN)

Application

EP 12700934 A 20120120

Priority

  • EP 11000501 A 20110121
  • EP 2012000259 W 20120120
  • EP 12700934 A 20120120

Abstract (en)

[origin: WO2012098006A1] The present invention relates to methods for the identification of HD AC interacting compounds using the ligand having the structure wherein R is H, C1-C6 alkyl, or cycloalkyl and X is a C1-C6 alkyl, cycloalkyl or an aryl, wherein the ligand is immobilized on a solid support via the NHR-group as well as to compounds having said structures.

IPC 8 full level

C12Q 1/34 (2006.01); C07C 259/00 (2006.01); G01N 33/68 (2006.01)

CPC (source: EP)

C07C 259/06 (2013.01); C12Q 1/34 (2013.01); G01N 33/6848 (2013.01); G01N 2333/98 (2013.01)

Citation (search report)

See references of WO 2012098006A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DOCDB simple family (publication)

WO 2012098006 A1 20120726; EP 2665829 A1 20131127

DOCDB simple family (application)

EP 2012000259 W 20120120; EP 12700934 A 20120120