EP 2665829 A1 20131127 - COMPOUNDS AND METHODS FOR THE IDENTIFICATION AND CHARACTERIZATION OF HDAC INTERACTING COMPOUNDS
Title (en)
COMPOUNDS AND METHODS FOR THE IDENTIFICATION AND CHARACTERIZATION OF HDAC INTERACTING COMPOUNDS
Title (de)
VERBINDUNGEN UND VERFAHREN ZUR IDENTIFIKATION UND CHARAKTERISIERUNG VON HDAC-INTERAGIERENDEN VERBINDUNGEN
Title (fr)
COMPOSÉS ET PROCÉDÉS POUR L'IDENTIFICATION ET LA CARACTÉRISATION DE COMPOSÉS INTERAGISSANT AVEC L'HDAC
Publication
Application
Priority
- EP 11000501 A 20110121
- EP 2012000259 W 20120120
- EP 12700934 A 20120120
Abstract (en)
[origin: WO2012098006A1] The present invention relates to methods for the identification of HD AC interacting compounds using the ligand having the structure wherein R is H, C1-C6 alkyl, or cycloalkyl and X is a C1-C6 alkyl, cycloalkyl or an aryl, wherein the ligand is immobilized on a solid support via the NHR-group as well as to compounds having said structures.
IPC 8 full level
C12Q 1/34 (2006.01); C07C 259/00 (2006.01); G01N 33/68 (2006.01)
CPC (source: EP)
C07C 259/06 (2013.01); C12Q 1/34 (2013.01); G01N 33/6848 (2013.01); G01N 2333/98 (2013.01)
Citation (search report)
See references of WO 2012098006A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
DOCDB simple family (application)
EP 2012000259 W 20120120; EP 12700934 A 20120120