Global Patent Index - EP 2683696 A1

EP 2683696 A1 20140115 - PROCESS FOR MAKING CRYSTALLINE FORM A OF LINEZOLID

Title (en)

PROCESS FOR MAKING CRYSTALLINE FORM A OF LINEZOLID

Title (de)

VERFAHREN ZUR HERSTELLUNG EINER KRISTALLINEN FORM VON LINEZOLID

Title (fr)

PROCÉDÉ DE PRÉPARATION DE LA FORME CRISTALLINE A DU LINÉZOLID

Publication

EP 2683696 A1 20140115 (EN)

Application

EP 11707846 A 20110309

Priority

EP 2011053555 W 20110309

Abstract (en)

[origin: WO2012119653A1] The invention relates to a process for making crystalline linezolid Form A, comprising a step of dissolving linezolid in an organic solvent at a temperature of at least 80°C to obtain a solution followed by a step of precipitation, said step preferably comprising adding, upon maintaining the temperature of at least 80°C, an antisolvent to said solution in an amount sufficient to induce precipitation of linezolid.

IPC 8 full level

C07D 263/20 (2006.01)

CPC (source: EP)

C07D 263/20 (2013.01)

Citation (search report)

See references of WO 2012119653A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DOCDB simple family (publication)

WO 2012119653 A1 20120913; EP 2683696 A1 20140115

DOCDB simple family (application)

EP 2011053555 W 20110309; EP 11707846 A 20110309