EP 2708537 A1 20140319 - HETEROAROMATIC RING DERIVATIVE
Title (en)
HETEROAROMATIC RING DERIVATIVE
Title (de)
HETEROAROMATISCHES RINGDERIVAT
Title (fr)
DÉRIVÉ À CYCLE HÉTÉROAROMATIQUE
Publication
Application
Priority
- JP 2011105188 A 20110510
- JP 2012061745 W 20120508
Abstract (en)
The compound represented by formula (IA) or a pharmaceutically acceptable salt thereof is based on orexin (OX) receptor antagonist activity, is useful in the treatment and prevention of illnesses including sleep disorder, depression, anxiety disorder, panic disorder, schizophrenia, drug dependency, Alzheimer's disease, Parkinson's disease, Huntington's chorea, eating disorders, pain, gastrointestinal disease, epilepsy, inflammation, immunological disease, endocrinological related disease, and hypertension.
IPC 8 full level
C07D 401/14 (2006.01); A61K 31/4192 (2006.01); A61K 31/422 (2006.01); A61K 31/4245 (2006.01); A61K 31/4439 (2006.01); A61K 31/506 (2006.01); A61P 1/00 (2006.01); A61P 5/00 (2006.01); A61P 9/12 (2006.01); A61P 25/08 (2006.01); A61P 25/16 (2006.01); A61P 25/20 (2006.01); A61P 25/22 (2006.01); A61P 25/24 (2006.01)
CPC (source: EP US)
A61P 1/00 (2018.01 - EP); A61P 3/04 (2018.01 - EP); A61P 5/00 (2018.01 - EP); A61P 9/12 (2018.01 - EP); A61P 25/00 (2018.01 - EP); A61P 25/04 (2018.01 - EP); A61P 25/08 (2018.01 - EP); A61P 25/14 (2018.01 - EP); A61P 25/16 (2018.01 - EP); A61P 25/18 (2018.01 - EP); A61P 25/20 (2018.01 - EP); A61P 25/22 (2018.01 - EP); A61P 25/24 (2018.01 - EP); A61P 25/28 (2018.01 - EP); A61P 25/30 (2018.01 - EP); A61P 29/00 (2018.01 - EP); A61P 29/02 (2018.01 - EP); A61P 37/00 (2018.01 - EP); C07D 401/14 (2013.01 - EP US); C07D 403/12 (2013.01 - EP US); C07D 413/12 (2013.01 - EP US); C07D 413/14 (2013.01 - EP US)
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
EP 2708537 A1 20140319; EP 2708537 A4 20141001; JP WO2012153729 A1 20140731; TW 201249830 A 20121216; US 2014081025 A1 20140320; WO 2012153729 A1 20121115
DOCDB simple family (application)
EP 12781685 A 20120508; JP 2012061745 W 20120508; JP 2013514014 A 20120508; TW 101116659 A 20120510; US 201214115933 A 20120508