EP 2710010 A1 20140326 - NOVEL CRYSTALLINE SALTS OF ASENAPINE
Title (en)
NOVEL CRYSTALLINE SALTS OF ASENAPINE
Title (de)
NEUE KRISTALLINE ASENAPINSALZE
Title (fr)
NOUVEAUX SELS CRISTALLINS D'ASÉPINE
Publication
Application
Priority
- EP 11166312 A 20110517
- EP 2012058964 W 20120515
- EP 12721519 A 20120515
Abstract (en)
[origin: EP2524921A1] The present invention relates to novel crystalline salts of Asenapine and to methods of their preparation. In particular, the invention relates to crystalline Asenapine salts of tartaric acid or succinic acid, wherein the salts are e.g. selected from the group consisting of Asenapine D, L-tartrate hydrate form A, Asenapine D, L-tartrate hydrate form B, Asenapine D, L-tartrate anhydrous form , Asenapine succinate form X, Asenapine succinate form , and Asenapine succinate form II. Furthermore the present invention relates to pharmaceutical compositions comprising the novel salts and to the novel salts for use in the treatment of psychotic diseases or disorders.
IPC 8 full level
A61K 31/407 (2006.01); A61P 25/18 (2006.01); C07D 491/044 (2006.01)
CPC (source: EP US)
A61K 31/407 (2013.01 - EP US); A61P 25/18 (2017.12 - EP); C07D 491/044 (2013.01 - EP US); C07D 491/22 (2013.01 - US)
Citation (search report)
See references of WO 2012156384A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
DOCDB simple family (publication)
EP 2524921 A1 20121121; EP 2710010 A1 20140326; US 2014163083 A1 20140612; WO 2012156384 A1 20121122
DOCDB simple family (application)
EP 11166312 A 20110517; EP 12721519 A 20120515; EP 2012058964 W 20120515; US 201214116098 A 20120515