Global Patent Index - EP 2776400 A1

EP 2776400 A1 20140917 - SUBSTITUTED PYRAZOLYL-BASED CARBOXAMIDE AND UREA DERIVATIVES BEARING A PHENYL MOIETY SUBSTITUTED WITH A CO-CONTAINING GROUP AS VANILLOID RECEPTOR LIGANDS

Title (en)

SUBSTITUTED PYRAZOLYL-BASED CARBOXAMIDE AND UREA DERIVATIVES BEARING A PHENYL MOIETY SUBSTITUTED WITH A CO-CONTAINING GROUP AS VANILLOID RECEPTOR LIGANDS

Title (de)

SUBSTITUIERTE CARBOXAMIDE AUF PYRAZOLUYLBASIS UND HARNSTOFFDERIVATE MIT EINEM MIT EINER CO-HALTIGEN GRUPPE SUBSTITUIERTEN PHENYLTEIL ALS VANILLOID-REZEPTORLIGANDEN

Title (fr)

DÉRIVÉS DE CARBOXAMIDE ET D'URÉE À BASE DE PYRAZOLYLE SUBSTITUÉ PORTANT UN FRAGMENT PHÉNYLE REMPLACÉ PAR UN GROUPE CONTENANT CO COMME LIGANDS DES RÉCEPTEURS VANILLOÏDES

Publication

EP 2776400 A1 20140917 (EN)

Application

EP 12781344 A 20121108

Priority

  • EP 11008926 A 20111109
  • EP 2012072146 W 20121108
  • EP 12781344 A 20121108

Abstract (en)

[origin: WO2013068467A1] The invention relates to substituted pyrazolyl-based carboxamide and urea derivatives bearing a phenyl moiety substituted with a CO-containing group as vanilloid receptor ligands, to pharmaceutical compositions containing these compounds and also to these compounds for use in the treatment and/or prophylaxis of pain and further diseases and/or disorders.

IPC 8 full level

C07D 231/12 (2006.01); A61K 31/415 (2006.01); A61P 29/00 (2006.01)

CPC (source: EP)

A61P 1/00 (2017.12); A61P 1/04 (2017.12); A61P 1/12 (2017.12); A61P 3/04 (2017.12); A61P 7/00 (2017.12); A61P 9/10 (2017.12); A61P 9/12 (2017.12); A61P 11/00 (2017.12); A61P 11/06 (2017.12); A61P 11/14 (2017.12); A61P 13/02 (2017.12); A61P 13/10 (2017.12); A61P 15/10 (2017.12); A61P 17/00 (2017.12); A61P 17/04 (2017.12); A61P 17/06 (2017.12); A61P 19/02 (2017.12); A61P 19/10 (2017.12); A61P 21/00 (2017.12); A61P 25/00 (2017.12); A61P 25/06 (2017.12); A61P 25/08 (2017.12); A61P 25/14 (2017.12); A61P 25/16 (2017.12); A61P 25/24 (2017.12); A61P 25/28 (2017.12); A61P 25/30 (2017.12); A61P 25/32 (2017.12); A61P 25/36 (2017.12); A61P 27/02 (2017.12); A61P 29/00 (2017.12); A61P 31/22 (2017.12); A61P 37/08 (2017.12); A61P 43/00 (2017.12); C07D 231/12 (2013.01)

Citation (search report)

See references of WO 2013068467A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2013068467 A1 20130516; EP 2776400 A1 20140917; JP 2014532746 A 20141208; KR 20140091042 A 20140718

DOCDB simple family (application)

EP 2012072146 W 20121108; EP 12781344 A 20121108; JP 2014540458 A 20121108; KR 20147015422 A 20121108