Global Patent Index - EP 2788352 A1

EP 2788352 A1 20141015 - AMORPHOUS FORM OF SITAGLIPTIN SALTS

Title (en)

AMORPHOUS FORM OF SITAGLIPTIN SALTS

Title (de)

AMORPHE FORM VON SITAGLIPTIN-SALZEN

Title (fr)

FORME AMORPHE DE SELS DE SITAGLIPTINE

Publication

EP 2788352 A1 20141015 (EN)

Application

EP 12816517 A 20121207

Priority

  • IN 3577DE2011 A 20111208
  • IB 2012057086 W 20121207

Abstract (en)

[origin: WO2013084210A1] The present invention claims amorphous solid state forms of sitagliptin salts, processes for their preparation, and pharmaceutical compositions thereof. As salt forming anions are claimed: The maleate, fumarate, besylate, mesylate and succinate. (Formula (I))

IPC 8 full level

C07D 487/04 (2006.01); A61K 31/4985 (2006.01); A61P 3/10 (2006.01)

CPC (source: EP US)

A61P 3/10 (2017.12 - EP); C07D 487/04 (2013.01 - EP US)

Citation (search report)

See references of WO 2013084210A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

DOCDB simple family (publication)

WO 2013084210 A1 20130613; WO 2013084210 A9 20131121; EP 2788352 A1 20141015; US 2014350023 A1 20141127

DOCDB simple family (application)

IB 2012057086 W 20121207; EP 12816517 A 20121207; US 201214363959 A 20121207