Global Patent Index - EP 2908802 A1

EP 2908802 A1 20150826 - A SOLID ORAL PHARMACEUTICAL FORMULATION CONTAINING TICAGRELOR

Title (en)

A SOLID ORAL PHARMACEUTICAL FORMULATION CONTAINING TICAGRELOR

Title (de)

FESTE ORALE PHARMAZEUTISCHE FORMULIERUNG MIT TICAGRELOR

Title (fr)

FORMULATION PHARMACEUTIQUE ORALE SOLIDE CONTENANT DU TICAGRÉLOR

Publication

EP 2908802 A1 20150826 (EN)

Application

EP 13792574 A 20131015

Priority

  • CZ 2012705 A 20121016
  • CZ 2013000130 W 20131015

Abstract (en)

[origin: WO2014059955A1] The present solution provides a solid oral pharmaceutical formulation containing ticagrelor, in the chemical name (1S,2S,3R,5S)-3-[7-[[(1R,2S)-2-(3,4-difluorophenyl)cyclopropyl]amino]- 5-(propylthio)-3H-1,2,3-triazolo[4,5-d]pyrimidin-3-yl]-5-(2-hydroxyethoxy)-1,2- cyclopentanediol, comprising at least one non-hygroscopic filler and/or at least one non- hygroscopic binder, wherein neither the filler, nor the binder have any disintegration effect. Preparation of the formulation is possible by wet granulation or dry granulation or direct

IPC 8 full level

A61K 9/00 (2006.01); A61K 9/20 (2006.01)

CPC (source: EP)

A61K 9/2018 (2013.01); A61K 9/2054 (2013.01); A61K 9/2095 (2013.01); A61K 9/2866 (2013.01); A61P 9/00 (2017.12); A61P 9/10 (2017.12)

Citation (search report)

See references of WO 2014059955A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2014059955 A1 20140424; BR 112015008076 A2 20170704; CN 104661649 A 20150527; CZ 2012705 A3 20140423; EA 201590745 A1 20150831; EP 2908802 A1 20150826; HK 1205456 A1 20151218; IL 238036 A0 20150531; IL 238036 B 20190530; JP 2015533129 A 20151119; JP 6301934 B2 20180328; KR 20150067153 A 20150617; MX 2015003866 A 20150717; UA 116784 C2 20180510; ZA 201501954 B 20170426

DOCDB simple family (application)

CZ 2013000130 W 20131015; BR 112015008076 A 20131015; CN 201380050404 A 20131015; CZ 2012705 A 20121016; EA 201590745 A 20131015; EP 13792574 A 20131015; HK 15106027 A 20150624; IL 23803615 A 20150330; JP 2015535983 A 20131015; KR 20157007818 A 20131015; MX 2015003866 A 20131015; UA A201504754 A 20131015; ZA 201501954 A 20150320