EP 2934502 A1 20151028 - PROCESS FOR PREPARARING N-(2-(7-METHOXY-1-NAPHTHALENYL)ETHYL) ACETAMIDE AND SOLID FORMS THEREOF
Title (en)
PROCESS FOR PREPARARING N-(2-(7-METHOXY-1-NAPHTHALENYL)ETHYL) ACETAMIDE AND SOLID FORMS THEREOF
Title (de)
VERFAHREN ZUR HERSTELLUNG VON N-(2-(7-METHOXY-1-NAPHTHALENYL)ETHYL)ACETAMID UND FESTE FORMEN DAVON
Title (fr)
PROCÉDÉ DE PRÉPARATION DE N-(2-(7-MÉTHOXY-1-NAPHTALÉNYL)ÉTHYL)ACÉTAMIDE ET DE FORMES SOLIDES DE CELUI-CI
Publication
Application
Priority
- EP 12199081 A 20121221
- EP 13153338 A 20130130
- EP 2013077725 W 20131220
- EP 13821818 A 20131220
Abstract (en)
[origin: WO2014096373A1] The present invention refers to solid forms of agomelatine, a process for their preparation and pharmaceutical compositions containing them. The present invention also relates to a process for the manufacture of N-[2-(7-methoxy- -naphthalenyl) ethyl]acetamide (agomelatine) with improved yields and purity and reducing the steps of the global process.
IPC 8 full level
A61K 31/165 (2006.01); A61P 25/00 (2006.01); C07C 233/18 (2006.01)
CPC (source: EP)
A61K 31/165 (2013.01); A61P 25/00 (2017.12); C07C 53/18 (2013.01); C07C 233/18 (2013.01); C07B 2200/13 (2013.01)
Citation (search report)
See references of WO 2014096373A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
DOCDB simple family (application)
EP 2013077725 W 20131220; EP 13821818 A 20131220