Global Patent Index - EP 2934502 A1

EP 2934502 A1 20151028 - PROCESS FOR PREPARARING N-(2-(7-METHOXY-1-NAPHTHALENYL)ETHYL) ACETAMIDE AND SOLID FORMS THEREOF

Title (en)

PROCESS FOR PREPARARING N-(2-(7-METHOXY-1-NAPHTHALENYL)ETHYL) ACETAMIDE AND SOLID FORMS THEREOF

Title (de)

VERFAHREN ZUR HERSTELLUNG VON N-(2-(7-METHOXY-1-NAPHTHALENYL)ETHYL)ACETAMID UND FESTE FORMEN DAVON

Title (fr)

PROCÉDÉ DE PRÉPARATION DE N-(2-(7-MÉTHOXY-1-NAPHTALÉNYL)ÉTHYL)ACÉTAMIDE ET DE FORMES SOLIDES DE CELUI-CI

Publication

EP 2934502 A1 20151028 (EN)

Application

EP 13821818 A 20131220

Priority

  • EP 12199081 A 20121221
  • EP 13153338 A 20130130
  • EP 2013077725 W 20131220
  • EP 13821818 A 20131220

Abstract (en)

[origin: WO2014096373A1] The present invention refers to solid forms of agomelatine, a process for their preparation and pharmaceutical compositions containing them. The present invention also relates to a process for the manufacture of N-[2-(7-methoxy- -naphthalenyl) ethyl]acetamide (agomelatine) with improved yields and purity and reducing the steps of the global process.

IPC 8 full level

A61K 31/165 (2006.01); A61P 25/00 (2006.01); C07C 233/18 (2006.01)

CPC (source: EP)

A61K 31/165 (2013.01); A61P 25/00 (2017.12); C07C 53/18 (2013.01); C07C 233/18 (2013.01); C07B 2200/13 (2013.01)

Citation (search report)

See references of WO 2014096373A1

Designated contracting state (EPC)

AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR

Designated extension state (EPC)

BA ME

DOCDB simple family (publication)

WO 2014096373 A1 20140626; EP 2934502 A1 20151028

DOCDB simple family (application)

EP 2013077725 W 20131220; EP 13821818 A 20131220