EP 2953456 A4 20160720 - TETRACYCLIC HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HEPATITIS C
Title (en)
TETRACYCLIC HETEROCYCLE COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HEPATITIS C
Title (de)
TETRACYCLISCHE HETEROCYCLISCHE VERBINDUNGEN SOWIE VERFAHREN ZUR VERWENDUNG DAVON ZUR BEHANDLUNG VON VIRENERKRANKUNGEN
Title (fr)
COMPOSÉS HÉTÉROCYCLIQUES TÉTRACYCLIQUES ET LEURS PROCÉDÉS D'UTILISATION POUR LE TRAITEMENT DE L'HÉPATITE C
Publication
Application
Priority
- CN 2013000128 W 20130207
- US 2014014361 W 20140203
Abstract (en)
[origin: WO2014121416A1] The present invention relates to compounds of formula (I) that are useful as hepatitis C virus (HCV) NS5B polymerase inhibitors, the synthesis of such compounds, and the use of such compounds for inhibiting HCV NS5B polymerase activity, for treating or preventing HCV infections and for inhibiting HCV viral replication and/or viral production in a cell-based system.
IPC 8 full level
A61K 31/397 (2006.01); C07D 471/04 (2006.01); C07D 471/14 (2006.01); C07D 471/20 (2006.01); C07D 471/22 (2006.01); C07D 487/14 (2006.01); C07D 519/00 (2006.01)
CPC (source: EP US)
A61K 31/4375 (2013.01 - EP US); A61K 31/438 (2013.01 - EP US); A61K 31/444 (2013.01 - EP US); A61K 31/4985 (2013.01 - EP US); A61K 31/5025 (2013.01 - EP US); A61K 31/519 (2013.01 - EP US); A61K 31/55 (2013.01 - EP US); A61K 45/06 (2013.01 - EP US); A61P 31/14 (2017.12 - EP); C07D 471/04 (2013.01 - EP US); C07D 471/14 (2013.01 - EP US); C07D 471/20 (2013.01 - EP US); C07D 471/22 (2013.01 - EP US); C07D 487/14 (2013.01 - EP US); C07D 519/00 (2013.01 - EP US)
C-Set (source: EP US)
Citation (search report)
- [I] US 2012328569 A1 20121227 - MCCOMAS CASEY CAMERON [US], et al
- [I] WO 2004041201 A2 20040521 - VIROPHARMA INC [US], et al
- See references of WO 2014123793A1
Designated contracting state (EPC)
AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR
Designated extension state (EPC)
BA ME
DOCDB simple family (publication)
WO 2014121416 A1 20140814; EP 2953456 A1 20151216; EP 2953456 A4 20160720; EP 2953456 B1 20190522; US 2015361101 A1 20151217; US 9243002 B2 20160126; WO 2014123793 A1 20140814
DOCDB simple family (application)
CN 2013000128 W 20130207; EP 14748737 A 20140203; US 2014014361 W 20140203; US 201414766462 A 20140203